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1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethan-1-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[2-(2-methylphenyl)ethyl]piperidine
(1R,7S)-3-[4-(2-hydroxyethyl)phenyl]-N-methyl-4-oxo-N-(pyrimidin-4-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-cyclopentyl-2-(3-{[methyl(oxolan-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
6-methyl-3-[(4-methyl-1H-imidazol-2-yl)methyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(thiophene-3-carbonyl)piperidine-2-carboxamide
N-[(4-cyanophenyl)methyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-2-oxo-2-phenylacetamide
2-[(4-ethylpiperazin-1-yl)methyl]-4-(6-methoxypyridin-2-yl)phenol
2-({2-[3-(dimethylamino)pyrrolidin-1-yl]acetamido}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-({1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}oxy)-N-(pyridin-4-ylmethyl)benzamide
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[3-(1H-pyrazol-1-yl)phenyl]methyl})amine
2-{2-[(1E)-pent-1-en-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-cyclohexyl-2-(2-oxo-1,2-dihydropyridin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
4-{[cyclopropyl({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl})amino]methyl}-2-methoxyphenol
N-[5-({[2-(dimethyl-1,3-thiazol-2-yl)ethyl]carbamoyl}amino)-2-methoxyphenyl]propanamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
3-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenol
(2S)-2-[1-benzyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]pyrrolidine-1-carboxamide
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
6-amino-1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]hexan-1-one
N-[4-(3-methoxyphenyl)phenyl]-4-(3-methoxypropyl)piperazine-1-carboxamide
4-(2,8-dimethylquinoline-3-carbonyl)-1-phenylpiperazin-2-one
6-{[(2,3-dimethyl-1H-indol-5-yl)methyl]amino}-N,N-dimethylpyridine-3-carboxamide
4-[1-(3-methylbutyl)-5-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
1-[2-(2,5-dimethylphenoxy)ethyl]-1-methyl-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]urea
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}ethan-1-one
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-[(methylsulfanyl)methyl]pyridine
1-(1,2-oxazole-3-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
1-(cyclohexylmethyl)-5-(thiomorpholine-4-carbonyl)piperidin-2-one
(3S,4S)-4-(morpholin-4-yl)-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-ol
N-(adamantan-1-yl)-3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
2-[(2S)-2-aminopropanoyl]-N-(cyclopropylmethyl)-N-propyl-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N4-[2-(benzyloxy)ethyl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
N-methyl-2-[3-(methylsulfanyl)phenyl]-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
2-{3-[2-(methylsulfanyl)ethyl]-5-[(propan-2-yloxy)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
{1-[(5-ethylfuran-2-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidin-4-yl}methanol
N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-(pyridin-2-ylmethyl)-4-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
9-(2-propoxypropanoyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(3-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-chloro-N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]benzamide
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
methyl 3-ethyl-2-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-3H-imidazo[4,5-b]pyridine-6-carboxylate
3-[2-(4-aminopiperidin-1-yl)-2-oxoethyl]-1-benzyl-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-chloro-4-[4-methyl-6-(methylamino)pyrimidin-2-yl]benzamide