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3-(1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)pyridine
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)imidazo[1,2-a]pyrimidine-2-carboxamide
4,5-dimethyl-6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
methyl (2S,4R)-1-[(3,4-difluorophenyl)methyl]-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
1-ethyl-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
N-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-tert-butyl-1-methyl-1H-pyrazole-5-carboxamide
2-cyclopropyl-N-[2-(dimethylamino)ethyl]-N-ethylpyrimidine-5-carboxamide
N-[(3S,5S)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
methyl 1-benzyl-5-{[(3-methoxyphenyl)methyl]amino}-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(2-ethylphenyl)-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,4-diazepan-5-one
5-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
N-(1-carbamoylcyclopentyl)-6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
8-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-(2-methoxyethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{5-[1-(methoxymethyl)cyclopropyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl}-3-methylpyridine
methyl 1-methyl-5-{[2-(pyridin-2-yl)piperidin-1-yl]sulfonyl}-1H-pyrrole-2-carboxylate
N-methyl-N-[3-(piperidin-1-yl)propyl]piperidin-3-amine
7-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
4-[4-(oxolan-2-ylmethyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-(thiophen-2-ylmethyl)piperidine
(4aR,8aS)-1-(2,5-difluorobenzoyl)-N,N-dimethyl-decahydro-1,6-naphthyridine-6-sulfonamide
(3S,7S)-5-(4,4,4-trifluorobutanoyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetamide
ethyl 4-[(2R,3R)-2-hydroxy-3-(2-phenylacetamido)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]piperidine-1-carboxylate
5-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-N,N-dimethylpyrimidin-2-amine
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
methyl 5-{[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]carbamoyl}-1-methyl-1H-pyrazole-3-carboxylate
N-(2,5-dimethylphenyl)-N'-(2-phenoxyethyl)propanediamide
5-methoxy-2-[3-(5-methylfuran-2-yl)-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl]-1,4-dihydropyridin-4-one
2-cyclopropyl-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyrimidin-4-ol
N-[1-(4-methanesulfonylphenyl)propyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
1-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-3-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]urea
(2R,3R,6R)-5-cyclobutanecarbonyl-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-benzofuran-2-carboxamide
1-cyclohexyl-N-[1-(pyrazin-2-yl)propan-2-yl]piperidine-4-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
1-[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1'-(5-hydroxypyridine-2-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
3-[3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]pyridine
5-(2-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]amino}pyrimidin-4-yl)-2-ethoxybenzoic acid
2-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
3-chloro-4-hydroxy-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]benzamide
3-methyl-1-(1-{6-[(thiophen-3-ylmethyl)amino]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
[2-(prop-2-en-1-yloxy)-5-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl]methanol
2-{[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
1-methyl-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine-2-carboxylic acid