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(3S,4S)-4-methyl-1-(5,6,7,8-tetrahydronaphthalene-2-carbonyl)piperidine-3,4-diol
1-(2-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrimidin-4-yl)piperidin-4-ol
2-(3-methylbut-2-en-1-yl)-8-(2-methylpyridin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
ethyl (4aS,8aR)-6-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylate
2-amino-N-{1-[(3-chlorophenyl)amino]-2-methylpropan-2-yl}-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
7-{[2-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}-1H-indole
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
8-(oxolane-3-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
4-[5-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]pyridin-2-amine
6-{4-[(2,2-dimethyloxan-4-yl)methyl]piperazin-1-yl}-9H-purine
(2S,4S)-4-{4-[4-(azepan-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxylic acid
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-(morpholin-3-yl)acetamide
7-(3-methoxypropyl)-2-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(piperidin-3-ylmethyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-1,2,3-triazole-4-carboxamide
methyl 3-{[1,5-bis(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
N-ethyl-5-(2-fluorophenyl)-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
8-(8-chloro-2-methylquinoline-4-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-methyl-1H-indole
N-benzyl-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}propanamide
1-[3-(dimethylamino)propyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(3R,5S)-5-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyrrolidin-3-ol
1-[2-(4-fluorophenyl)ethyl]-4-{[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amino}pyrrolidin-2-one
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-(pyrimidin-4-ylmethyl)acetamide
N,N-bis(1,3-oxazol-4-ylmethyl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
methyl 6-cyclobutyl-2-[(cyclohexylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}ethyl)-1,2,3,4-tetrahydrophthalazine-1,4-dione
4-({3-[(2R,5S)-2,5-dimethylpyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)morpholine
2-(2-phenylethyl)-9-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(3S)-N,N-dimethyl-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]azepan-3-amine
6-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]pyrimidin-4-amine
6-{1-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]piperidin-4-yl}pyrimidin-4-ol
{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-[(2-fluorophenyl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-oxo-N-(propan-2-yl)piperidine-3-carboxamide
N-[2-({2-[(4-chlorophenyl)methyl]-1,3-benzoxazol-5-yl}formamido)ethyl]acetamide
2-{[4-(2-methoxy-5-methylphenyl)-5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}-N-[(2-methoxyphenyl)methyl]-8-methylquinazolin-4-amine
4-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1-methylimidazolidin-2-one
N-({8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)pyridine-3-carboxamide
1-(3-{4-[(dimethylamino)methyl]phenyl}phenyl)propan-1-one
2-cyclopropyl-5-{4-[(2-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-3,4-dihydropyrimidin-4-one
N-({4-hydroxy-1-[4-(trifluoromethyl)benzoyl]azepan-4-yl}methyl)cyclopropanecarboxamide
(2S)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
2,7-dimethyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
4-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-1-cyclopentylpiperazin-2-one
3-[(3R,4S)-1-{2-[methyl(phenyl)amino]acetyl}-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
4-(5-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
5-[3,5-bis(trifluoromethyl)phenyl]pyrazin-2-amine
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[4-(2-methylpyridin-4-yl)-1H-pyrazol-1-yl]acetamide