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(4aS,8aR)-1-butyl-6-[2-(pyrazin-2-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
2-methyl-5-propyl-4-(2,3,4-trimethoxyphenyl)pyrimidine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-6-methylpyridazin-3-amine
2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-propyl-1H-imidazole
2-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-ol
4-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}morpholine
2-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1,3-thiazole-4-carboxamide
N-(1-{2-oxo-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
5-[4-(1-methoxyethyl)phenyl]-2-(propan-2-yl)-1,3-thiazole
methyl(quinolin-6-ylmethyl){[4-(2-{4-[4-(trifluoromethyl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl}amine
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-[(5-methylthiophen-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
4-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-2-methylquinoline
N2-benzyl-6-(pyrimidin-5-yl)-1,3,5-triazine-2,4-diamine
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
N-[1-(3-chlorophenyl)cyclopropyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
4-(4-hydroxycyclohexyl)-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
2-cyclopropyl-N-[2-(1H-imidazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N,N-dimethyl-2-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-sulfonamide
4-cyclopentyl-7-(2,3-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(2S)-1-methoxypropan-2-yl]-4-{[(2S)-pyrrolidin-2-ylmethyl]sulfamoyl}benzamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-methoxyethyl)-N-(propan-2-yl)benzamide
6-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-9H-purine
1-(2-ethylpyrimidine-5-carbonyl)-4-phenylpiperidine-4-carbonitrile
4-methyl-6-{4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]piperidin-1-yl}pyrimidin-2-amine
4-[2-({[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)ethyl]phenol
1-(2H-1,3-benzodioxol-5-yl)-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methylpiperidin-4-amine
(2S)-4-methyl-1-(oxolan-2-ylmethyl)-2-(propan-2-yl)piperazine
4-[7-(3-methoxypiperidin-1-yl)pyrazolo[1,5-a]pyrimidin-5-yl]pyridine
N-[3-(cyclohexylsulfanyl)propyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-2-(1H-indazol-3-yl)ethan-1-one
(3aR,6aR)-2-(2-hydroxyethyl)-5-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-1λ6-thiomorpholine-1,1-dione
8-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
4-(furan-3-ylmethyl)-3-{2-[4-(4-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
2-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methylacetamido]acetamide
9-(cyclopropylmethyl)-4-(1H-imidazol-2-ylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(4aS,8aR)-1-(4-hydroxybutyl)-6-[2-(methylsulfanyl)acetyl]-decahydro-1,6-naphthyridin-2-one
[2-(4-methoxyphenoxy)ethyl]({[6-(trifluoromethyl)pyridin-3-yl]methyl})amine
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(morpholin-4-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(2-methoxybenzoyl)piperazin-1-yl]propan-1-one
1-(5-ethyl-1,2-oxazole-3-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
5-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-cyclopentyl-4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-methyl-1-{[3-(pyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}-1H-1,3-benzodiazole
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-(2-phenylethyl)piperazin-2-yl]ethan-1-ol
2-(2,5-dimethoxyphenyl)-8-methyl-3-[(4-methylpiperazin-1-yl)methyl]quinoline
5-chloro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyridine-2-carboxamide
N-{[3-(cyclopentyloxy)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-3-carboxamide