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1-(4-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}-1,4-diazepan-1-yl)ethan-1-one
3-{[methyl(prop-2-en-1-yl)amino]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
[5-(1-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-1H-imidazol-2-yl)furan-2-yl]methanol
8-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(3,5-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-fluoropyridine-2-carbonyl)piperidin-3-ol
3-(dimethylamino)-N-[(2-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)benzamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]quinoline-2-carboxamide
8-(6-carboxypyrimidin-4-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3,5-dimethoxy-N-({1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}methyl)benzamide
4-(2-methoxyphenoxy)-1-{spiro[2.3]hexane-1-carbonyl}piperidine
N-[(2,6-difluorophenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
5-(3-fluorophenoxymethyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-3-carboxamide
1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
7-(2-methoxyethyl)-2-[3-(1H-pyrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decane
1-(pyridin-4-ylmethyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
2-(oxolan-2-ylmethyl)-9-[3-(pyridin-4-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
4-benzyl-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(1H-pyrrole-2-carbonyl)piperazine
1-[3-(cyclopentyloxy)phenyl]-3-methyl-3-[1-(1,2-oxazol-3-yl)ethyl]urea
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-3-[5-(4-methylphenyl)furan-2-yl]propan-1-one
7-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[2-(dimethylamino)ethyl]-5-oxo-N-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-3-carboxamide
5-{[methyl(thiophen-3-ylmethyl)amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
1-{5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
2-(2-hydroxyethyl)-9-(6-methylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2S)-oxolane-2-carbonyl]-4-phenoxypiperidine-4-carboxylic acid
4-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
dimethyl[(3-{7-methyl-2,7-diazaspiro[4.4]nonane-2-carbonyl}phenyl)methyl]amine
1-[3-(1H-imidazol-1-yl)phenyl]ethan-1-ol
(1R,7S)-3-(2-methoxyethyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-[3-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)phenoxy]acetamide
7-(8-hydroxyquinoline-7-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-methyl-2-(1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
(1-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-2-yl)methanol
[1-(1,3-benzothiazol-2-ylmethyl)-4-[(3-methoxyphenyl)methyl]piperidin-4-yl]methanol
6-{[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]amino}-N,N-dimethylpyridine-3-carboxamide
{4-[5-(morpholine-4-carbonyl)pyridin-2-yl]-1,4-oxazepan-6-yl}methanol
1-(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-[2-(2-phenoxyethoxy)phenyl]-2-(pyridin-4-ylsulfanyl)acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(2-phenylpropyl)-1H-1,2,3-triazole
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(pyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{[3-(4-hydroxyphenyl)phenyl]formamido}-N-methylbutanamide
2-{4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-5-methyl-4-(thiophen-2-yl)pyrimidine
1-[(2-chloro-4-fluorophenyl)methyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(3-hydroxypiperidin-1-yl)ethan-1-one
4-{1-[1-(4-chlorophenyl)cyclobutanecarbonyl]piperidin-4-yl}morpholine
1-{5-[(4-ethylpiperazin-1-yl)methyl]-2-methoxyphenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
2-{[(1,4-dimethyl-1H-pyrazol-5-yl)methyl](methyl)amino}-1-phenylethan-1-ol