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1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(3-methoxybenzoyl)piperazine
N-{3-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}-4-fluorobenzamide
2-ethoxy-5-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}pyridine
8-(1-benzothiophen-2-ylmethyl)-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3R,4S)-1-(2-methoxypyridine-4-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
(3S)-N-tert-butyl-2-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
3-{1-[3-(1H-imidazol-1-yl)propanoyl]piperidin-4-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-7-methylquinolin-3-yl}methanol
1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
N-(2-methoxyethyl)-4-methyl-2-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3-thiazole-5-carboxamide
1-cyclopentyl-N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
4-(1-methyl-1H-pyrazol-4-yl)-1-(3-phenylpropyl)-1,2,3,6-tetrahydropyridine
2-[2-(4-{2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)ethoxy]ethan-1-ol
N-{1-[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
{1-[6-(dimethylamino)pyrazin-2-yl]-3-[(4-fluorophenyl)methyl]piperidin-3-yl}methanol
4-(2-methoxy-6-methylbenzoyl)-2-(4-methylpentyl)morpholine
2,6-dimethoxy-3-[2-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]pyridine
1-{2-[(1-methyl-5-phenyl-1H-pyrrol-2-yl)formamido]ethyl}piperidine-3-carboxamide
2-{6-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
N-(2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-2-methylpropanamide
2-methoxy-N-{1-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
9-[(2,4-difluorophenyl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
6-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
4-methyl-6-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]pyrimidin-2-amine
4-[1-(1-methyl-1H-indole-4-carbonyl)piperidin-3-yl]benzoic acid
N-[(3-chloropyridin-4-yl)methyl]-N-(pyridin-3-ylmethyl)cyclopropanamine
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-[(2,6-dimethylphenyl)amino]propan-1-one
3-[(4-acetamidopiperidin-1-yl)methyl]-N-(1,2,4-thiadiazol-5-yl)benzamide
6-[(3-methoxyphenyl)methoxy]-4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
N-[(3S,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-(4-cyclohexylpiperazin-1-yl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
2-{3-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-ylmethyl]-6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline
6-methoxy-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidin-4-amine
5-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrazine-2-carboxamide
1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
5-(1H-imidazol-5-yl)-3-(1-phenylcyclopropyl)-1,2,4-oxadiazole
3-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}thiophene-2-carboxamide
(3R,4R)-1-(8-methoxyquinolin-2-yl)-4-(morpholin-4-yl)piperidin-3-ol
(2S,4R)-4-amino-1-(3,4-dimethoxybenzoyl)-N-ethylpyrrolidine-2-carboxamide
4-{1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}thiomorpholine
2-(dimethyl-1,3-thiazol-5-yl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-(1,2-oxazol-5-yl)-4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenol
1-[(diethylcarbamoyl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
5-{2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[(dimethylcarbamoyl)amino]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
5-[2-methyl-4-(4-methylphenyl)-5-oxopiperazine-1-carbonyl]pyridine-2-carbonitrile
2,8-dimethyl-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]quinoline-4-carboxamide