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1-{5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]thiophen-2-yl}ethan-1-one
butyl 1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
8-[5-(morpholin-4-ylmethyl)pyridin-2-yl]quinoline
(3aR,6aS)-2-[1-(2-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-octahydropyrrolo[3,4-c]pyrrole
N-(3-ethyl-4-methyl-1H-pyrazol-5-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-1-cyclohexylpiperidine-4-carboxamide
1-[(1-{6-[methyl(2-methylpropyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-(1-propylpiperidin-4-yl)ethyl]methylamine
2-amino-4-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3-benzothiazole-6-carboxamide
5-(azepane-1-carbonyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-ethyl-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidine-3-carboxylic acid
4-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-3,4-dihydroquinazoline-2-carboxamide
4-[(3,5-dimethoxyphenyl)methyl]-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetamide
2-methyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidine
2-{2-methyl-3-[({[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}amino)methyl]-1H-indol-1-yl}acetamide
N-benzyl-2-[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]acetamide
1-[(3,4-dimethylphenyl)methyl]-4-(hydroxymethyl)azepan-4-ol
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethyl-1,3-oxazole-4-carboxamide
3-{[3-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-N-(1,2-oxazol-5-ylmethyl)benzamide
methyl 3-[4-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-6-[(3-methoxyphenyl)methoxy]-2-oxo-1,4-diazepan-1-yl]propanoate
ethyl 5-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
(2R,3R,6R)-5-(1H-1,3-benzodiazole-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2-hydroxyphenyl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-pyrazole-5-carboxamide
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(2-phenylethyl)piperidine
6-cyclohexanecarbonyl-N-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
2,4-dimethyl-6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyrimidine
2-(2,4-difluorophenoxy)-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyrrolidin-3-yl]methanesulfonamide
8-fluoro-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}quinoline-2-carboxamide
1-(1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-[(5-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(4-methoxypyrimidin-2-yl)pyrrolidin-3-yl]acetamide
5-ethyl-2-methyl-4-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}pyrimidine
(1R,5R)-6-(cyclobutylmethyl)-3-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
[4-({4-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)phenyl]methanol
N-methyl-1-[1-(3-phenylpropyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3-(1H-1,2,3-benzotriazol-1-yl)propan-1-one
3-(naphthalene-1-carbonyl)piperidine
8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-4-phenyl-9-(pyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecane
1-{3-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]phenyl}imidazolidin-2-one
N-cyclopropyl-5-(4-methanesulfonylphenyl)thiophene-2-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
2-methoxy-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]pyridine-3-carboxamide
N-phenyl-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine