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4-(1,4-dithiepan-6-yl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-benzyl-4-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-1,4-diazepan-6-ol
5-methyl-2-phenyl-4-[4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazol-5-yl]-1,3-oxazole
2-(3-hydroxypiperidin-1-yl)-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
(2S,4R)-1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-N-(2-methylpropyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4,5-dimethyl-6-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]pyrimidin-2-amine
2-(5-cyano-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)-N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-one
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-N-(3-fluorophenyl)piperidin-3-amine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[1-(2-chlorophenyl)ethyl]propanamide
3-{5-[2-(1H-imidazol-2-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-(4-fluorophenyl)-1-[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
4-methoxy-N-({1-[2-(pyrrolidin-1-yl)acetyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
N-(2-fluorophenyl)-3-[1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(pyridin-3-yl)ethan-1-one
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-(4-{[5-(2,3-dichlorophenyl)furan-2-yl]methyl}morpholin-3-yl)acetic acid
1-(4-fluorophenyl)-4-[1-(2-methoxyethyl)piperidine-4-carbonyl]-1,4-diazepane
7-methyl-2-(1-phenylcyclopentanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{2-[7-(2,6-dimethylhept-5-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methoxybenzamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-2-(1H-pyrazol-1-yl)acetamide
1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
3-ethyl-8-(2,3,4,9-tetrahydro-1H-carbazole-8-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-methoxy-N-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]-4-(prop-2-en-1-yl)piperidine-1-carboxamide
N-ethyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
2-{5-[1-(ethylsulfanyl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}pyridine
3-methyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-(1-methyl-1H-pyrazole-4-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N3-cyclooctyl-4-oxo-N5-(prop-2-en-1-yl)-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-(2,4,5-trimethylphenyl)-1,2,4,5,10,11-hexaazatricyclo[7.3.0.02,6]dodeca-3,5,7,9,11-pentaene
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(4-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}({[4-(methylsulfanyl)phenyl]methyl})(pyridin-4-ylmethyl)amine
2-(methylsulfanyl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
3-hexyl-8-[2-(morpholin-2-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N2-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-N1-(pyridin-3-yl)ethane-1,2-diamine
4-(3-aminoazepane-1-carbonyl)-5,6,7,8-tetrahydroquinazolin-2-amine
N-benzyl-2-(2-methyl-5-oxopyrrolidin-1-yl)-N-(2,2,2-trifluoroethyl)acetamide
2-methyl-4-({4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}methyl)-1,3-thiazole
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-phenylpyrimidine-5-carboxamide
(2R)-2-amino-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-methylpentanamide
3,5-dimethyl-N-[2-(4-propylmorpholin-2-yl)ethyl]-1,2-oxazole-4-sulfonamide
4-{[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(3S,4R)-1-[2-(2,3-dihydro-1H-isoindol-2-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
4-(2-{1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-2-yl}ethyl)phenol
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(2-methoxyphenyl)-2-methylpiperazine