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6-[2-(isoquinolin-5-yl)-1H-imidazol-1-yl]-2-methylheptan-2-ol
{[(1R,5S,6R)-3-cyclopropanecarbonyl-3-azabicyclo[3.1.0]hexan-6-yl]methyl}(prop-2-en-1-yl)(pyridin-2-ylmethyl)amine
2-benzyl-8-(6-methylpyridazin-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
N4-[2-(2-fluorophenoxy)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-(2-methylpropyl)-4-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]pyrrolidin-3-yl}piperidine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-6-methoxypyrimidin-4-amine
(1S,5R)-6-(pyridin-2-ylmethyl)-3-(quinolin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
5-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)-2,3-dihydro-1H-pyrazol-3-one
N-(2-methoxyethyl)-4-[3-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(2,3-dimethylphenyl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[(1-methyl-1H-indol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
9-[(2-ethylpyrimidin-5-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S)-2-oxoazepan-3-yl]-4-(4-{[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}piperidin-1-yl)benzamide
methyl 3-{[3-(azepane-1-carbonyl)-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
1-[2-(piperazin-1-yl)ethyl]-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1-{3-[(trimethylpyrimidin-4-yl)amino]propyl}piperidin-3-yl)methanol
4-methyl-2-({1-methyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-1,2-dihydrophthalazin-1-one
5-acetyl-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]thiophene-2-carboxamide
4-chloro-3-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]-1H-pyrazol-5-amine
1-[1-(1-benzylpiperidin-4-yl)piperidine-3-carbonyl]-1,4-diazepan-5-one
(2R)-N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methoxy-2-phenylacetamide
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-4-methylpentan-1-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-(2-methoxyacetyl)-N-methylpiperidine-4-carboxamide
N-(pyridin-2-ylmethyl)-4-[4-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(5-acetylthiophen-3-yl)-N-methyl-N-[2-(4-methylpiperidin-1-yl)ethyl]acetamide
2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-{[7-fluoro-5-(quinolin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(3R,9aR)-8-[(2,4-dimethylphenyl)methyl]-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[3-(4-methanesulfonylphenyl)phenyl]-5-methyl-1,3,4-thiadiazole
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-{[3-(methylsulfanyl)phenyl]methyl}benzamide
1-{1'-[(3-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-(2-phenylethyl)piperidine-1-carboxamide
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methylaniline
N2-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-N4-ethylpyrimidine-2,4-diamine
N-butyl-1-cyclohexyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
1-ethyl-2-oxo-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,2-dihydropyridine-4-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-5-(methoxymethyl)-N-methylthiophene-2-carboxamide
1-cyclohexyl-4-(3-methylbut-2-en-1-yl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-cyclopropyl-4-{[4-(2-methylphenyl)phenyl]methyl}piperazine-2-carboxamide
N-cyclooctyl-2-{4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}acetamide
N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-(2-{7-[(2,3-difluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)acetamide
1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
1-(4-cyclopentyl-1,4-diazepan-1-yl)-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-cycloheptyl-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl}acetamide
1-{2-[4-(3-phenylpiperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}piperazine
(3R,4R)-4-amino-1-[4-(4-propylphenyl)benzoyl]piperidin-3-ol
9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one