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1,3-dimethyl-6-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-2-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(pyridin-3-ylmethyl)piperidin-3-amine
[(3R,4R)-1-[1-(4-fluorophenyl)piperidin-4-yl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
9-(2,3-dihydroxybenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}cyclobutanecarboxamide
N-{2-[1-(4-fluorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
N-[(2-aminopyrimidin-5-yl)methyl]-N,2,7,8-tetramethylquinoline-4-carboxamide
1-{2-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]ethyl}pyrrolidin-2-one
N-methyl-1-(2-methylpropyl)-5-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]pyrrolidine-3-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidine
N,2,6-trimethyl-N-[1-(1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
3-(4-fluorophenyl)-N-(2-hydroxy-2-phenylethyl)-1H-pyrazole-5-carboxamide
5-[2-(3-methoxy-4-methylphenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[5-(3-methylphenyl)-1H-indol-1-yl]acetamide
2-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-(4H-1,2,4-triazol-4-yl)piperidine
N-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carboxamide
(3S,4S)-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidine-3,4-diol
5-methoxy-2-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}-4H-pyran-4-one
4-[(2-fluorophenyl)methyl]-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
5-(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)pyrazin-2-amine
4-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-6-fluoro-1,2,3,4-tetrahydroquinolin-2-one
4-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
(3aS,7aR)-2-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-[(2R,3R,6R)-5-(1-ethyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-5-methylthiophene-2-carboxamide
8-methyl-4-(piperidine-1-carbonyl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline
(2S,4R)-4-amino-N,N-diethyl-1-(2,6,8-trimethylquinoline-4-carbonyl)pyrrolidine-2-carboxamide
4-{[3-(cyclopentyloxy)phenyl]methyl}thiomorpholine
[(3R,4R)-1-(1,3-benzoxazol-2-yl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(5-methoxy-1-methyl-1H-indole-2-carbonyl)piperidine-4-carboxylic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-cyclopropylpyrimidine-5-carboxamide
4-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(2R,3S,6R)-3-(4-fluorophenyl)-5-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-methoxyphenyl)-5-(3-methyl-1,2-oxazol-5-yl)-1H-1,2,4-triazole
1-(4-{4-[2-(3,4-dimethylphenyl)-1H-imidazol-1-yl]phenyl}piperazin-1-yl)ethan-1-one
1-(2-aminoethyl)-N-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(4-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]acetic acid
(1R,3S)-3-[1-(5-chloro-2-methoxyphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]cyclopentan-1-amine
1-[2-(1-benzylpiperidin-2-yl)ethyl]-3-(6-chloropyridin-3-yl)urea
4,5-dimethyl-2-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]-1,3-thiazole
2,3-dimethyl-6-[2-(naphthalen-2-yloxy)propanoyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
3-{5-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
(2R,3R)-3-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-(thiophen-3-yl)piperidine-1-carboxamide
1-{4-[4-(4-cyclopentylpiperazine-1-carbonyl)-2-methoxyphenoxy]piperidin-1-yl}ethan-1-one
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine