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2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N,N-dimethyl-2-[(1S,5R)-6-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-(2-methyl-1-{7-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)pyridine-2-carboxamide
1-[phenyl(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-1,2,3,4-tetrazole
1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
ethyl 5-[2-(4-fluorophenyl)morpholin-4-yl]pentanoate
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-[(3R,4R)-1-[(5-butylthiophen-2-yl)methyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
5-[3-(4-methylbenzenesulfonyl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(cyclopropylmethyl)-6-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}pyrrolidin-2-one
N,N-dimethyl-2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-2-phenylacetamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(pyrrolidine-3-carbonyl)piperidine
2-[(3,5-difluorophenyl)methyl]-8-(oxolan-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
1-{4-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-4-oxobutyl}piperidin-2-one
3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-5-methyl-1,2,4-oxadiazole
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-(5-ethyl-2-methylpyrimidin-4-yl)-N-methylpiperidin-4-amine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(2-phenylethyl)pyrrolidin-3-yl]-5-methyl-1,2-oxazole-4-carboxamide
N-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-methyl-5-(5-propylpyrimidin-2-yl)quinoline
methyl 6-benzyl-2-{[2-(2-fluorophenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(4-{[2-(benzylamino)pyrimidin-5-yl]methyl}-1,4-oxazepan-6-yl)methanol
{[2-(azocan-1-yl)pyridin-3-yl]methyl}[(3-fluoro-4-methoxyphenyl)methyl]amine
4-[(5-{1-[2-(ethylsulfanyl)ethyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
methyl 4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
3-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
5,5-dimethyl-3-(2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
1-(cyclohexylmethyl)-N3-ethyl-4-oxo-N5-[2-(pyridin-4-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-ethoxy-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyrimidine
(3S,9aR)-3-ethyl-8-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-ethyl-N-[(1-methanesulfonylpiperidin-3-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-(2-fluoro-6-methoxyphenyl)-1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-1H-imidazole
1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-4-oxo-2-propyl-N-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-{[6-oxo-2-(thiophen-2-yl)-1,6-dihydropyrimidin-4-yl]methyl}acetamide
1-[2-(3-fluorophenyl)ethyl]-N-methyl-N-(1-methylpiperidin-4-yl)-6-oxopiperidine-3-carboxamide
(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl](4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-methyl-1-(thiophen-3-ylmethyl)urea
7-{3-[5-(4-methylphenyl)furan-2-yl]propanoyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
5-[5-(furan-3-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-[(4-methyl-1H-imidazol-5-yl)methyl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
6-(cyclopentylamino)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
2-fluoro-N-{3-[(pyridin-3-yl)amino]propyl}-5-sulfamoylbenzamide
3-fluoro-N-{1-[1-(3-methoxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-6-methyl-4H-pyran-4-one
(1R,2S)-2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}cyclopentan-1-ol
2-(cyclopropylmethyl)-8-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-(3-cyanophenyl)-5-{1-[2-(methylsulfanyl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-(4-chloro-1H-pyrazole-3-carbonyl)-3,9-diazaspiro[5.5]undecane
2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]pyridine-3-carbonitrile