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7-[2-(benzyloxy)ethyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-ethyl-3-methoxybenzamide
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(5-methylfuran-2-yl)methyl]amine
1-(3,5-dichloro-4-methylbenzoyl)-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
1-cyclohexanecarbonyl-N-[1-(1H-pyrazol-1-yl)propan-2-yl]pyrrolidine-2-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
7-(1-benzothiophen-3-yl)-4-(3-methoxybenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-[(4-fluoro-2-methoxyphenyl)methyl]-[1,2,4]triazolo[4,3-a]pyridin-3-amine
3-[(dimethylcarbamoyl)methyl]-1-[(4-fluorophenyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-ethyl-N-[(4-fluorophenyl)methyl]-2-methanesulfonylacetamide
ethyl 4-(2-phenylethyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-4-carboxylate
N-({1-[(2-cyanophenyl)methyl]piperidin-3-yl}methyl)-2-methoxyacetamide
1-[3-(cyclohexylsulfanyl)propyl]-3-(3-methylcinnolin-5-yl)urea
(2E)-N-[(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-3-[2-(methylsulfanyl)pyrimidin-5-yl]prop-2-enamide
8-[(3-hydroxyphenyl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-{[4-(trifluoromethoxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-{[(1R,2S,5R)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl]methyl}-5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carboxamide
1-(5-acetyl-2-ethoxyphenyl)-3-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]urea
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-({1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}carbamoyl)pyridin-1-ium-1-olate
5-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
2-{4-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]phenyl}acetamide
2-methoxy-5-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
1-(2-chlorobenzoyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridine
N-ethyl-3,3,3-trifluoro-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)propanamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-ethyl-N,4-dimethyl-1,3-thiazole-5-carboxamide
(3R)-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}pyrrolidin-3-ol
2-{4-[(6-chloro-2H-chromen-3-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(2-oxopyrrolidin-3-yl)-1,3-oxazole-4-carboxamide
6-[2-(methylsulfanyl)benzoyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
5-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-(3-methyl-4-{[8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-[2-(2-oxopiperidin-1-yl)ethyl]urea
4,6-dimethyl-2-oxo-N-[4-(pyridin-2-yl)butyl]-1,2-dihydropyridine-3-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
(1R,5R)-6-benzyl-3-(2,4-dimethylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
8-(3-methylbut-2-en-1-yl)-1-oxa-8-azaspiro[4.6]undecan-9-one
2-methoxy-1-(4-methyl-2-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}piperazin-1-yl)ethan-1-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5-ethyl-1,3,4-oxadiazol-2-amine
5-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-1,2-oxazol-3-ol
4-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}-2-methoxyphenol
2-(4-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-amido}-3,5-dimethyl-1H-pyrazol-1-yl)acetic acid
1-(2-methoxyacetyl)-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-4-carboxamide
N-{1-[1-(2-acetylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
3-[(2-{7,9-dioxo-8-azaspiro[4.5]decan-8-yl}acetamido)methyl]-4-methylbenzoic acid
5-methoxy-N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]furan-2-carboxamide
4-{4-[6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carbonyl]-2-oxopiperazin-1-yl}benzonitrile