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6-chloro-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]imidazo[1,2-a]pyridine-2-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-4-(pyridin-3-yl)pyrimidin-2-amine
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)methanesulfonamide
4-[2-(2-hydroxyphenoxy)acetyl]-1-(3-methoxyphenyl)piperazin-2-one
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
4-[(2R,3R)-1'-benzoyl-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperazin-2-one
1-{1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]piperidin-4-yl}pyrrolidin-2-one
4-oxo-4-[2-(pyridin-2-yl)pyrrolidin-1-yl]butane-1-sulfonamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(thian-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(2-aminopyrimidin-5-yl)-N-cycloheptyl-7-fluoroquinoline-4-carboxamide
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)oxan-4-amine
1-[3-(2-fluorophenoxy)azetidin-1-yl]-2-(pyridin-3-yloxy)ethan-1-one
4-{[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]methyl}-N-(1-methyl-1H-pyrazol-4-yl)benzamide
N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]propanamide
[1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-yl]methanol
N2,N2,5,6-tetramethyl-N4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrimidine-2,4-diamine
methyl 3-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}benzoate
3-[2-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(cyclohexyloxy)-3-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propan-2-ol
1-[2-(azepan-1-yl)-2-phenylethyl]-3-(1,3-dimethyl-1H-pyrazol-4-yl)urea
5-({[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(5-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
2-{3-[3-(dimethylamino)phenyl]phenoxy}acetamide
1-[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]-2-(pyridin-4-yl)ethan-1-one
3-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
N-tert-butyl-2-methyl-3-[2-(pyridin-3-yloxy)acetamido]benzamide
[1-(quinolin-4-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
1-{3-[3-(3-methylphenoxy)azetidine-1-carbonyl]piperidin-1-yl}propan-1-one
5-(3-methylquinolin-2-yl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)acetamide
2-{4-[6-(dimethylamino)pyrimidin-4-yl]phenyl}acetic acid
1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-4-(1,3-thiazol-2-yl)piperazine
1-(azepan-1-yl)-3-(2-methoxy-4-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
5-acetyl-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}thiophene-3-carboxamide
(1S,5R)-6-propyl-3-{2-[3-(trifluoromethyl)phenyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-benzyl-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-N-methylpiperidin-3-amine
2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]pyridine-3-carbonitrile
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-5,6-dimethylpyrimidin-4-amine
{4-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]phenyl}methanol
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)acetamide
4-methyl-1-[3-(1-methyl-1H-imidazole-2-carbonyl)phenyl]-1H-pyrazole
4-{2-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}-1-(propan-2-yl)pyrrolidin-2-one
methyl N-[1-({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)ethyl]carbamate
6-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]hexan-1-ol
(4aR,7aS)-4-[2-(2,4-dimethylphenoxy)ethyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propane-1,2-diol
1-(1,2-benzoxazol-6-yl)-3-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)urea
dimethyl[({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}methyl)sulfamoyl]amine
1-cyclohexyl-3-(cyclopropylmethyl)-N-(2-hydroxyethyl)-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide