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N-cyclobutyl-1-cyclopropyl-6-oxopiperidine-3-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-{[2-(dimethylamino)pyridin-3-yl]methyl}acetamide
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
5-methyl-3-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-indole-2-carboxylic acid
6-(dimethylamino)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyridine-3-carboxamide
[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)(quinolin-3-ylmethyl)amine
N-[4-(2-fluorophenoxy)phenyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine-4-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[(3-methyl-1-benzofuran-2-yl)methyl]acetamide
2-(4-ethoxyphenyl)-6,7-dimethoxyquinazolin-4-amine
3-cyclopropyl-1-(1H-indazol-6-yl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
3-methyl-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
8-[5-(morpholin-2-ylmethyl)-3-phenyl-1H-1,2,4-triazol-1-yl]quinoline
(3R,4R)-4-(4-methylpiperazin-1-yl)-1-(6-phenylpyridazin-3-yl)piperidin-3-ol
3-(azepane-1-carbonyl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
dimethyl({2-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-2-yl]ethyl})amine
4-(1H-indol-5-yl)thiophene-2-carboxylic acid
6-[3-(2-ethylphenoxy)azetidine-1-carbonyl]quinoline
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-4-carbonitrile
5-benzyl-1-(3-methoxyphenyl)-4-(1-methylcyclopropanecarbonyl)piperazin-2-one
3-[(2-fluorophenyl)formamido]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}propanamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)benzamide
dimethyl[(5-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}thiophen-3-yl)methyl]amine
(3R,4R)-4-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pyrrolidin-3-ol
dimethyl({[4-methyl-5-(1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
6-methyl-5-[5-(4-methyl-1,2,5-oxadiazol-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
3-{1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
5-{[4-(3-chloropyridin-2-yl)piperazin-1-yl]methyl}-2-(ethylsulfanyl)pyrimidine
4-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N,N-diethyl-1-[1-(quinolin-4-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
3-(3-ethylphenoxy)-1-(oxolane-3-carbonyl)azetidine
(1R,3R,5S)-3-(4-methoxyphenyl)-8-(2-methyl-1,3-thiazole-4-carbonyl)-8-azabicyclo[3.2.1]octane
3-(cyclopropylsulfamoyl)-5-(2-fluoro-3-methoxyphenyl)benzoic acid
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
4-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}piperazin-2-one
6-methoxy-3-{[4-(1-methylpiperidin-4-yl)piperidin-1-yl]methyl}-1H-indazole
1-{6-hydroxy-4-[(2-methyl-1-benzothiophen-3-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
N-[(3R,4S)-1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
2-ethyl-N-[2-(furan-2-yl)ethyl]-4-methyl-1,3-oxazole-5-carboxamide
2-(4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]-N-(oxolan-2-ylmethyl)propanamide
2-(2,5-dioxoimidazolidin-4-yl)-N-[2-(naphthalen-1-yl)propan-2-yl]acetamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
methyl (1R,3S,3aR,6aS)-3-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
7-(cyclohexylmethyl)-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(5-{[3-(morpholin-4-ylmethyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
(isoquinolin-5-ylmethyl)(methyl)[(1-phenyl-1H-pyrazol-5-yl)methyl]amine
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-2-methyl-4,5,6,7-tetrahydro-2H-indazole