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(2,1,3-benzoxadiazol-5-ylmethyl)[(3-chloro-4,5-dimethoxyphenyl)methyl]methylamine
5-{1-[2-(4-chlorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
9-[(2-fluoro-4-methylphenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[4-(1-phenyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetamide
3-(4-chlorophenyl)-5-cyclopentanecarbonyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-(2-fluorophenyl)-1-[4-(hydroxymethyl)piperidin-1-yl]-3-phenylpropan-1-one
2-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-indene-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline
N-(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
2-[1-(2-butyl-1,3-benzoxazole-5-carbonyl)piperidin-2-yl]ethan-1-ol
N-ethyl-3-(3-hydroxy-3-methylbutyl)-N-[(3S,4R)-4-hydroxyoxolan-3-yl]benzamide
2-methyl-1-[4-(3-methylphenoxy)piperidin-1-yl]-2-(morpholin-4-yl)propan-1-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
1-(3-{[3-(azocane-1-carbonyl)-1H-pyrazol-5-yl]methoxy}phenyl)ethan-1-one
N-methyl-2-(3-methyl-2-oxoimidazolidin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-[(4-methoxyphenyl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
ethyl 2-{[3-(4-phenylbenzoyl)piperidine-1-carbonyl]amino}acetate
5-{2-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
8-(1-benzofuran-2-ylmethyl)-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{5-[(2-methoxyphenyl)methyl]-1,2,4-oxadiazol-3-yl}pyridine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-(1-methoxypropan-2-yl)-1,2-oxazole-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(2-methoxyphenyl)ethan-1-one
1-ethyl-N-[(3-fluorophenyl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-5-oxo-1-phenyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-2,5-dihydro-1H-pyrazole-3-carboxamide
2-(1H-1,3-benzodiazol-2-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(4-methoxy-3-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-{1-[2-(pyridin-2-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}piperidin-1-yl)ethan-1-one
(1-{1-[2-(difluoromethoxy)benzoyl]piperidin-4-yl}ethyl)dimethylamine
methyl 3-[(3S,4R)-4-(morpholin-4-yl)-1-[(3-phenoxyphenyl)methyl]piperidin-3-yl]propanoate
N,6-dimethyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]urea
4-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
N-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
2-[5-(azepan-1-ylmethyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1,5-dimethyl-1H-indole-2-carboxamide
N-(2-methoxyethyl)-2-[(prop-2-en-1-yl)amino]-N-(thiophen-2-ylmethyl)benzamide
5-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1H-indole
2-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}benzonitrile
5-acetyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}thiophene-3-carboxamide
1-[4-phenyl-1-(quinolin-2-ylmethyl)piperidin-4-yl]ethan-1-one
4-[(4-fluorophenyl)methyl]-1-(5-hydroxypyrazine-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
5-[4-(1H-pyrazol-5-yl)phenyl]-2,3-dihydro-1H-indol-2-one
3-amino-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}thiophene-2-carboxamide
3-{benzyl[(5-tert-butyl-1H-pyrazol-3-yl)methyl]amino}-2-methylpropan-1-ol
5-{2-[5-(4-methylphenyl)furan-2-yl]ethyl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-{1-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]ethyl}morpholine
1-[3-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)phenyl]ethan-1-one