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ethyl 4-(2-phenylethyl)-1-(thian-4-yl)piperidine-4-carboxylate
1-{1-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]azetidin-3-yl}-1H-pyrazole
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
4-{1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]azetidin-3-yl}pyridine
N-[(2-methylphenyl)methyl]-6-oxo-N,1-bis(prop-2-en-1-yl)piperidine-3-carboxamide
1-ethyl-3-(2-methylpropyl)-N-[1-(thiophen-3-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
(1R,5R)-N,N-dimethyl-6-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
4-propyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidine-5-carboxamide
1-cycloheptyl-N-(2-methylpropyl)-6-oxopiperidine-3-carboxamide
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
4-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-1-ethylpyrrolidin-2-one
1-(2-ethoxyethyl)-N,3-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
(3S,4R)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
4-[4-({4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)phenyl]but-3-yn-1-ol
N-[(3S,5S)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]-1-propylpiperidin-4-amine
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-decahydro-2,7-naphthyridine-2-sulfonamide
4-[3-carboxy-6-(4-fluorophenyl)pyridin-2-yl]piperazine-2-carboxylic acid
2-(3-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
5-[({[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
1-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)butan-1-one
1-{4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}piperidine-3-carboxamide
8-(2,2-dimethylpropyl)-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[methyl({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}quinolin-8-ol
2-[6-methyl-2-oxo-4-(trifluoromethyl)-1,2-dihydropyridin-1-yl]-N-propylpropanamide
(1S,4S)-2-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-azabicyclo[2.2.1]heptane
ethyl 1-(cyclopropylmethyl)-5-(oxolane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-acetyl-N-{1,9-dioxaspiro[5.5]undecan-4-yl}benzamide
1-{2-[1-(cyclopropylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-4-fluorophenyl}-1H-pyrazole
4-(2,6-dimethylpyrimidine-4-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(1R,7S)-3-[4-(2-hydroxyethyl)phenyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-amino-6-{4-[(dimethylamino)methyl]thiophen-2-yl}-4-(3-ethyl-1,2-oxazol-5-yl)pyridine-3-carbonitrile
(1R,3S)-3-{[(2-chlorophenyl)methyl](2-methoxyethyl)carbamoyl}cyclopentane-1-carboxylic acid
N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]morpholine-2-carboxamide
3-(2-chlorophenyl)-1-[4-(hydroxymethyl)piperidin-1-yl]-3-phenylpropan-1-one
(3aR,6aR)-2-benzyl-N-(1H-1,2,4-triazol-5-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{4-[(4-methylphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-(5-methyl-2-pentanamidophenyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5,6-dimethyl-N-[2-(propan-2-ylsulfanyl)ethyl]pyridine-3-carboxamide
3-[(3R,4S)-1-[(4-chloro-2-fluorophenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propan-1-ol
N-methyl-N-(1-methylpyrrolidin-3-yl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
4-[4-(piperidine-1-carbonyl)phenoxy]-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine
4-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
(1R,9aR)-1-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-octahydro-1H-quinolizin-1-ol
8-(3,5-difluoropyridine-2-carbonyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(3-chloro-4-fluorophenyl)-3-cyclopropyl-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazole
N,N-dimethyl-4-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)piperidine-1-carboxamide
methyl (2S,4S,5R)-5-(4-chlorophenyl)-1,2-dimethyl-4-[methyl(oxan-4-yl)carbamoyl]pyrrolidine-2-carboxylate
1-({1-[3-(2-fluorophenyl)benzoyl]piperidin-4-yl}methyl)-4-methylpiperazine