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8-(1-benzothiophen-2-ylmethyl)-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-{4-[3-(benzylcarbamoyl)piperidin-1-yl]piperidin-1-yl}acetic acid
3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1-[3-(piperidin-1-ylmethyl)phenyl]urea
6-methyl-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-(oxan-4-yl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
2-[4-({methyl[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)piperidin-1-yl]ethan-1-ol
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(4,7,8-trimethylquinolin-2-yl)pyrrolidin-3-yl]methanol
9-(1-methyl-1H-pyrazole-4-carbonyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{[3-(difluoromethoxy)phenyl]methyl}-5-(4-methylpiperazin-1-yl)-2,3-dihydropyridazin-3-one
1-(2-{5-[(3Z)-hex-3-en-1-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)-4-methylpiperazine
2-phenyl-7-{spiro[2.3]hexane-1-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
9-(2-hydroxy-3-methylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(4aS,7aR)-1-[4-(dimethylamino)benzoyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(butan-2-yl)-1-ethyl-N-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(1H-pyrazol-1-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)benzamide
ethyl 4-{[2-(ethylamino)pyrimidin-5-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
4-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]phenol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
4-ethyl-1-methyl-3-[(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-1-benzothiophene-5-carboxamide
N-[(4-ethoxyphenyl)methyl]-4-methyl-5-(1-methyl-1H-pyrazol-3-yl)-1,3-thiazol-2-amine
(4aS,8aR)-1-(2-aminoethyl)-6-(2-cyclopentylacetyl)-decahydro-1,6-naphthyridin-2-one
3-[3-({[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
(4aS,7aR)-1-[(2-methoxyphenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(6-cyanopyridin-3-yl)-4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carboxamide
2-ethyl-N-{2-[4-(oxan-4-yl)morpholin-2-yl]ethyl}benzamide
N-ethyl-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(oxolan-2-ylmethyl)propanamide
(4aS,7aR)-1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}(2-methoxyethyl)(pyridin-2-ylmethyl)amine
N-[2-(ethylsulfanyl)ethyl]-7-fluoro-2-methylquinoline-4-carboxamide
N-benzyl-2-[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]acetamide
(5S,9aS,9bS)-5-(4-ethylphenyl)-2-(1-methylpiperidin-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
9-(4-methyl-1,3-thiazole-5-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-2-[(2-fluorophenyl)methyl]-5-(1-methyl-1H-pyrrole-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-methylphenol
5-{1-[(4-ethylphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,2,3-trimethylquinoxaline-6-carboxamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(1-benzothiophen-2-ylmethyl)-1-(cyclohexylmethyl)-N-methylpyrrolidine-2-carboxamide
N-methyl-2-[3-(pyridine-2-carbonyl)piperidin-1-yl]pyrimidin-4-amine
1-[(4-methyl-1H-imidazol-5-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
6-methoxy-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidin-4-amine
1-[4-(dimethylamino)azepan-1-yl]-4-(4-methoxyphenyl)butane-1,4-dione
N-{2-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propyl}cyclohexanecarboxamide
1-(1-{2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxybenzoyl}piperidin-3-yl)propan-1-one
3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-4-[(3-methoxyphenyl)methyl]piperazin-2-one