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N-{[4-(aminomethyl)phenyl]methyl}-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(2-oxopyrrolidin-1-yl)propanamide
N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-2-(methylamino)pyrimidine-5-carboxamide
1-methyl-4-[3-methyl-1-(3-methylbutyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
3-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-[3-(1H-pyrazol-4-yl)benzoyl]piperidine
1-(4-phenylbutyl)-4-(pyrimidin-2-yl)-1,4-diazepane
2-(5-acetylthiophen-3-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
({5-[1-(2,2-difluoroethyl)-1H-pyrazol-3-yl]thiophen-2-yl}methyl)[1-(6-methylpyridin-2-yl)propan-2-yl]amine
1,3-dimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-(3-{[(6-methoxy-2H-chromen-3-yl)methyl]amino}phenyl)-3-methylimidazolidin-2-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-4-ethyl-5-methylpyrimidin-2-amine
1-[4-(azepan-1-ylmethyl)-2-methoxyphenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
{[2-(butan-2-yloxy)-3-methoxyphenyl]methyl}[(5-methoxy-1H-indol-2-yl)methyl]amine
(1R,3S)-3-(2-aminoethoxy)-7-(naphthalene-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-6-(methoxymethyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2,1,3-benzoxadiazol-4-ylmethyl)-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
7-(2-methoxyethyl)-2-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
4-[(2,4-dimethoxyphenyl)methyl]-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]piperazin-2-one
2-amino-3-ethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(1H-1,2,4-triazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
11-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
2-[(4-methoxyphenyl)methyl]-N-(pyrimidin-4-ylmethyl)-1,3-benzoxazole-6-carboxamide
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
7-[5-(hydroxymethyl)furan-2-carbonyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[3-(1H-indazol-1-yl)propyl]-4-(trifluoromethyl)pyrimidin-2-amine
2-methyl-4-{4-[4-(1H-pyrrole-2-carbonyl)piperazine-1-carbonyl]phenyl}butan-2-ol
5-ethyl-N,2-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrimidin-4-amine
4-(2-{1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-2-yl}ethyl)phenol
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-(dimethylamino)-2-(4-fluorophenyl)-N-methylacetamide
3,5-dimethyl-1-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}pyrrolidin-3-yl)-1H-pyrazole
4-[(2S)-1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}pyrrolidine-2-carbonyl]morpholine
3-methyl-4-(1-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methylpyridin-2-amine
N-{3-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-3-oxopropyl}methanesulfonamide
6-{[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]methyl}pyridine-2-carboxylic acid
4-(3-oxo-3,4-dihydropyrazin-2-yl)-N-[2-(trifluoromethyl)phenyl]piperazine-1-carboxamide
5-cyclohexaneamido-1-(2-methoxyethyl)-N-[2-(2-methoxyphenyl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
2-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-3-methoxyphenol
N4-[(3S,4S)-1-ethyl-4-methoxypyrrolidin-3-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
14-[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-4-(thiophene-3-carbonyl)-1,4-diazepan-2-one
N-{2-[2-methyl-5-(morpholine-4-sulfonyl)-1H-1,3-benzodiazol-1-yl]ethyl}propanamide
1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-3-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
4,5-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)thiophene-2-carboxamide
methyl 4-{4-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]piperazin-1-yl}benzoate
6,8-dimethyl-2-({[2-(1-methylpyrrolidin-2-yl)ethyl]amino}methyl)quinolin-4-ol
2-amino-4-(2,4-dimethoxyphenyl)-6-(6-methoxypyridin-3-yl)pyridine-3-carbonitrile
[4-({methyl[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)oxan-4-yl]methanol