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1-methyl-4-({5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-ethyl-6-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyridine-2-carboxamide
1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
methyl 4-{[9-hydroxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
3-(2-chloro-4-fluoro-5-methylphenyl)-1-methyl-1-(piperidin-4-yl)urea
1-(2-aminoethyl)-N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
7-(1,2-oxazole-3-carbonyl)-N4-(oxolan-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]quinoxaline-5-carboxamide
1-(carbamoylmethyl)-N-[1-(3,5-difluorophenyl)cyclopropyl]piperidine-3-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[2-(1-methylpiperidin-3-yl)ethyl]propanamide
3-(2-methylpropyl)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1,2-oxazole-5-carboxamide
2-(cyclopentylmethyl)-1-(3-methoxypropyl)-6-methyl-3-[4-(4-methylphenyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
2-amino-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-(4-hydroxy-2-methoxyphenyl)pyridine-3-carbonitrile
(3S,4S)-1-[(5-methylfuran-2-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-(2-hydroxyethyl)-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-(2,1,3-benzoxadiazol-4-yl)-1-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5,7-dimethyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(1-phenylcyclopentanecarbonyl)piperidin-4-ol
2-(2-methylquinazolin-4-yl)benzamide
(3R,4R)-1-(2-ethoxypyridine-3-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
methyl 4-[5-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
(3aR,6aR)-2-[(3-chloropyridin-4-yl)methyl]-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N,2-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-{1-[1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
ethyl 3-({1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazol-4-yl}formamido)propanoate
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
4-{3-[(3S,4R)-3-acetamido-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]propoxy}benzamide
[({1-[(2-ethylphenyl)methyl]pyrrolidin-3-yl}methyl)sulfamoyl]dimethylamine
(3aR,6aR)-2-cyclopentyl-5-(thiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl (2S,4R)-4-(2,3-dimethyl-1H-indole-7-amido)-1-[(3-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
5-(2-{2,7-diazaspiro[4.5]decan-7-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
4-[(furan-2-ylmethyl)amino]-5-methyl-N-(3-phenylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
1-[2-(3-fluorophenyl)ethyl]-N-(oxan-4-yl)-6-oxopiperidine-3-carboxamide
1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-2-(1H-pyrazol-1-yl)ethan-1-one
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-[2-(phenylsulfanyl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(azepane-1-carbonyl)-1-ethyl-5-(morpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole
2-tert-butyl-6-(4-methanesulfonylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-(thiophen-2-yl)-4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
2-{4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(2-chloro-4-{[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl}-6-methoxyphenoxy)acetic acid
2,5-dimethyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
6-fluoro-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
2-[3-(2-aminoethyl)piperidine-1-carbonyl]benzene-1,3-diol
3-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N-(propan-2-yl)propanamide
N-(diphenylmethyl)-2-[2-(1-ethyl-3-oxopiperazin-2-yl)acetamido]acetamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-methyl-5-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
N3-butyl-N5-[3-(dimethylamino)-2,2-dimethylpropyl]-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
8-[2-(2-methoxyphenyl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid