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dimethyl(3-{2-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
2-(adamantan-1-yl)-5-(4-methoxypiperidine-1-carbonyl)pyrimidin-4-ol
{3-ethyl-1-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}methanol
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(5-methyl-1H-imidazol-4-yl)methyl]-1-[4-(propylsulfanyl)phenyl]urea
ethyl 2-(4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}morpholin-3-yl)acetate
(2-ethoxy-5-{[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenyl)methyl acetate
N-(3-phenylpropyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1H-1,2,4-triazole
2-amino-4-ethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1,3-thiazole-5-carboxamide
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-(1H-pyrazol-5-yl)piperidine
3-({[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]carbamoyl}(methyl)amino)-N-methylbutanamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}thian-4-amine
3-(2-methoxybenzenesulfonyl)-9-methyl-3,9-diazaspiro[5.6]dodecane
7-(1,3-benzothiazol-2-yl)-4-[(4-chlorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(cyclopropylmethyl)azepan-3-yl]-5-(1,2-oxazol-3-yl)thiophene-2-sulfonamide
1-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
2-{[5-(2-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}-2-methylpropanamide
(4S,4aS,8aR)-4-phenyl-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-decahydroquinolin-4-ol
1-[1-(2-ethylpyridine-4-carbonyl)piperidin-4-yl]piperidin-3-ol
1-{4-[2-(3,4-dimethoxyphenyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}pentane-1,4-dione
N-(1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperidin-4-yl)methanesulfonamide
8-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-1-oxa-8-azaspiro[4.5]decan-3-ol
1-methyl-2,4-dioxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
4-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-ethyl-3-methyl-1H-pyrazole
N-(1,2-diphenylethyl)-2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}acetamide
1-{2-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-(1-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
2-(4-fluorophenoxymethyl)-N-[2-(3-methylthiophen-2-yl)ethyl]-1,3-oxazole-4-carboxamide
4-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
3-(3-fluorophenyl)-4-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
1-benzyl-4-[(8-methoxyquinolin-2-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-(1-methyl-4-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
2-(2-aminoethyl)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]quinazolin-4-amine
4-{[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]methyl}benzonitrile
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-2-methylthieno[3,2-d]pyrimidin-4-amine
N-[3-(2-propoxyphenyl)propyl]oxane-2-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-5-methylpyrazine-2-carboxamide
2,6-dimethyl-N-{2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-4-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
5-(4-methoxyphenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
5-(1H-imidazol-2-ylmethyl)-2-(2-methoxyphenyl)-8-methyl-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-[3-({[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]carbamoyl}amino)-4-fluorophenyl]propanamide
5-methoxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}furan-2-carboxamide
N-(butan-2-yl)-N-(3-phenylprop-2-yn-1-yl)cyclopropanecarboxamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(oxolan-2-ylmethoxy)ethan-1-one
2-amino-4-({[1-(2-hydroxyethyl)piperidin-4-yl]methyl}(methyl)amino)quinazoline-6-carboxylic acid
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-cyclopropyl-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-[(3-aminopyrrolidin-1-yl)sulfonyl]-N-methyl-N-(1H-pyrazol-3-ylmethyl)benzamide