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1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(pyridin-3-yl)propan-1-one
5-amino-N-[(3S,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
N-ethyl-N-(pyridin-4-ylmethyl)-1-(thiophene-3-sulfonyl)piperidin-3-amine
N-[4-(2-fluorophenoxy)phenyl]-1-(furan-3-ylmethyl)piperidine-4-carboxamide
(1S,5R)-6-benzyl-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4,4,4-trifluoro-1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}butan-1-one
1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
4-fluoro-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
2-(3-phenylpropyl)-8-(pyrazine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(2E)-N-[(3-methyl-7-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(thiophen-2-yl)prop-2-enamide
8-(dimethyl-1,3-oxazole-5-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
3-{1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-methanesulfonyl-1,4-diazepane
4-{3-[(4aS,8aS)-decahydroisoquinoline-2-carbonyl]phenyl}-2-methylbutan-2-ol
2-methoxy-6-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)phenol
[3-(2-methoxyethyl)-1-(1H-pyrazole-3-carbonyl)piperidin-3-yl]methanol
1-{2-[1-(4-chloro-2-methylbenzoyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
4-chloro-3-[4-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-1H-pyrazol-5-amine
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
3-(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-4-yl)-1,3-oxazolidin-2-one
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
6,6-dimethyl-N-{3-[methyl(phenyl)amino]propyl}-5-oxothiomorpholine-3-carboxamide
3-(3-methoxypropyl)-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxylic acid
2-amino-4-(2-ethylpyrimidin-5-yl)-6-(3-methylphenyl)pyridine-3-carbonitrile
9-(5-acetylpyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
4-methoxy-6-(pyridin-4-yl)pyrimidin-2-amine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}benzamide
5-(propan-2-yl)-N-[1-(thian-4-yl)piperidin-4-yl]-1,2-oxazole-3-carboxamide
4-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)pyridin-2-amine
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-6-[2-(pyrrolidin-1-yl)ethyl]pyridine-3-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(3-hydroxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-methoxyphenoxy)-2-methyl-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
N-[(3S,4R)-1-(5-methylpyrazine-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
6-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
7-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
2-{5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl}acetic acid
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-1-ethyl-3,5-dimethyl-1H-pyrazole-4-carboxamide
5-(6-methoxypyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline
6-(2,5-dimethylfuran-3-yl)-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(pyrrolidin-1-yl)-2-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]ethan-1-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
2-[N-(3-methylphenyl)methanesulfonamido]-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidine
N4-[(2-methoxyphenyl)methyl]-2,N4-dimethylpyrimidine-4,6-diamine
(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl](1,3-thiazol-2-ylmethyl)amine
1-[(5-acetylthiophen-3-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidin-4-amine
1-[(2-chloro-5-fluorophenyl)methyl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine