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N-{4-[4-({imidazo[1,2-a]pyridin-2-ylmethyl}amino)piperidin-1-yl]phenyl}-3-phenylpropanamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)furan-3-carboxamide
2-[2-(benzyloxy)ethyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-ethoxy-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
5-(methoxymethyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyridine-2-carbonitrile
3-acetamido-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]butanamide
4-(5-ethylfuran-2-yl)-1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazole
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[3-(methylsulfanyl)propyl]acetamide
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-(hydroxymethyl)piperidin-3-ol
4-methyl-1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pentane-1,2-dione
4-(cyclobutylsulfamoyl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]benzamide
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-(2-phenylethyl)piperidine
1-(2-aminoethyl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(5,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl})methylamine
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-3-methylbutanamide
N-[2-(1-methylpiperidin-3-yl)ethyl]-1-propyl-1H-pyrazole-5-carboxamide
1-(3-hydroxyphenyl)-4-[1-(3-methylpyridin-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
1-{2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetyl}-N,N-diethylpiperidine-3-carboxamide
2-(4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-(2-hydroxyethyl)-N-{3-[methyl(phenyl)amino]propyl}-1H-1,3-benzodiazole-5-carboxamide
8-methyl-N-[(5-methylfuran-2-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[(2-chlorophenyl)methyl]-3-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}propanamide
3-(4-{[5-(3-chlorophenyl)furan-2-yl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
methyl 4-{4-[6-(1-hydroxyethyl)pyridin-2-yl]piperazin-1-yl}benzoate
N-(3-chloro-4-methylphenyl)-1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(propan-2-yloxy)propan-1-one
N3-[2-(cyclohex-1-en-1-yl)ethyl]-N5-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-2-yl}ethan-1-ol
2-[(3-chlorophenyl)methyl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,3-benzoxazole-6-carboxamide
2-[2-methyl-3-({[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}methyl)-1H-indol-1-yl]acetamide
6-[2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanoyl]-2-methyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]({4-[(dimethylamino)methyl]phenyl}methyl)methylamine
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}acetamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-ethylphenyl)methyl]-N-methylacetamide
methyl 4-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}pentanoate
1-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
4-{4-[(3,4-dimethoxyphenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-chloro-N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-6-fluoro-3-methylbenzamide
[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
5-(morpholin-4-ylmethyl)-N-(pyridin-2-ylmethyl)furan-3-carboxamide
3-(4-chlorophenyl)-1-(1H-imidazol-4-ylmethyl)piperidine
4-methyl-2-[1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
N-[3-(1H-imidazol-1-yl)propyl]-1-methyl-N-(pyridin-3-ylmethyl)azepane-2-carboxamide
N-[phenyl(pyridin-4-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
2-{2-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
N-(1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide