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3-acetamido-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
(4aR,8aS)-1-(3-methylthiophene-2-carbonyl)-6-(pyridine-2-carbonyl)-decahydro-1,6-naphthyridine
4-phenyl-N-[3-(4-{[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]butanamide
N-[4-(methylamino)butyl]-5-phenyl-1,2-oxazole-4-carboxamide
3-(4-hydroxyphenyl)-4-[2-(4-methoxyphenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopentyl-4-(4-{[2-hydroxy-3-(3-methoxyphenoxy)propyl]amino}piperidin-1-yl)benzamide
1-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]piperidine-2-carboxamide
N'1-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}cyclopropane-1,1-dicarboxamide
1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-ethyl-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
2-{2-methylimidazo[1,2-a]pyridin-3-yl}-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}acetamide
ethyl 4-[(5S,9aS,9bS)-2-(1-methylpiperidin-4-yl)-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]-1H-pyrazole-3-carboxylate
6-(4-cyclopentyl-1,4-diazepan-1-yl)-N-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-{1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(4-methyl-1H-imidazole-5-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[3-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazine-1-carbonyl)phenyl]methyl}dimethylamine
2-[(4-methoxyphenyl)methyl]-N-[(6-methylpyridin-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(1-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl]methanol
2-[4-(2-amino-9H-purin-6-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
(2E)-3-(3-fluorophenyl)-1-[4-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
2-(4-{[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
3-[3-(2H-1,3-benzodioxol-5-yl)phenyl]-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazole
5-acetyl-N-ethyl-2,4-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrrole-3-carboxamide
2-({[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
6-ethyl-N-[3-(4-methylbenzenesulfonamido)propyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
5-{3-[4-(furan-2-carbonyl)piperazin-1-yl]-3-oxopropyl}-5-[(4-phenylphenyl)methyl]pyrrolidin-2-one
3-methyl-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-phenylpiperidine
3-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
2-amino-6-(2,3-dihydro-1-benzofuran-5-yl)pyrimidin-4-ol
4-(azonan-1-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
5-{2-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
2-methyl-N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-5-(propan-2-yl)furan-3-carboxamide
7-methoxy-3-({methyl[2-(morpholin-4-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-[4-(3-fluoropyridin-2-yl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
2-[(2,4,5-trimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-methyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]azepane-2-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
(1R,3S)-7-(3-fluoro-4-methoxybenzoyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-(pyrrolidin-1-yl)-3-[5-(1,3-thiazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propan-1-one
8-{5-[(4-chloro-1H-pyrazol-1-yl)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}quinoline
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2,3,6-trimethylphenoxy)ethan-1-one
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-{[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4-methyl-1H-imidazole
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-5-cyclopropyl-N-methyl-1,2-oxazole-3-carboxamide
2-(2,2-dimethylpropanoyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-(2,6-dimethylpyridin-3-yl)-N-[1-(1H-imidazol-2-yl)ethyl]pyrimidin-2-amine
S-[2-(dimethyl-1,2-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-hydroxybutane-1-sulfonamido
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
3,5-dimethoxy-2-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)benzoic acid
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine