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3-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-N,N-dimethylpropane-1-sulfonamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2,3-dihydro-1,2-benzothiazol-3-one
3-(furan-2-yl)-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]propan-1-one
(2S,4R)-4-amino-N-[(5-methoxy-1H-indol-2-yl)methyl]pyrrolidine-2-carboxamide
4-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
2-amino-4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
6-(2-chlorophenyl)-2-(3-{[methyl(propan-2-yl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
[(2S,4R,5R)-5-(2-fluorophenyl)-1-methyl-4-({[1-(pyridin-2-ylmethyl)piperidin-4-yl]amino}methyl)pyrrolidin-2-yl]methanol
1-[2-({[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]piperidin-4-ol
4-[(2-methylphenyl)methyl]-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
5-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
4-ethyl-5-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-1,3-thiazol-2-amine
1-(1,4-dioxan-2-ylmethyl)-5-(4-fluoro-2-methylphenyl)-4-phenyl-1H-imidazole
N-methyl-3-{[(3-methylthiophen-2-yl)methyl]amino}-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
cyclopentyl 4-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)carbamoyl}amino)benzoate
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(1-ethylpiperidin-4-yl)acetamide
(4S)-N-[2-chloro-5-(trifluoromethyl)phenyl]-4-hydroxy-3,3,4-trimethylpiperidine-1-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
(3S,4R)-4-methyl-1-(2-methyl-1,3-thiazole-4-carbonyl)-3-(2-methylpropyl)piperidin-4-ol
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(pyridin-4-yl)acetamide
2-[2-({ethyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)phenoxy]acetic acid
7-(2-hydroxyethyl)-2-[(3-methylquinoxalin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-({5-[(2-phenoxyethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)propanamide
2-{methyl[2-(morpholin-4-yl)propyl]amino}pyridine-4-carboxamide
2-(4-ethoxyphenyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
(3R,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
2-methoxy-5-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyrimidine
2-methoxy-5-({methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amino}methyl)benzoic acid
4-(piperazine-1-sulfonyl)-N-{2-[(2R)-pyrrolidin-2-yl]ethyl}benzamide
N-(butan-2-yl)-N-[(4-chlorophenyl)methyl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
2-(5-acetylthiophen-3-yl)-N-[2-(1H-indol-1-yl)ethyl]-N-methylacetamide
methyl 2-(tert-butylsulfamoyl)-6-[(3-chlorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 2-(5-{1-[2-(cyclopent-2-en-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetate
2-[(4,5-dimethylfuran-2-yl)methyl]-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)propanamide
1,3-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-amino-4-(3,4-dihydroxyphenyl)-6-(propan-2-yl)pyridine-3-carbonitrile
N-methyl-N-(propan-2-yl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]pyrrolidin-3-amine
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-1-(4-hydroxypiperidin-1-yl)propan-1-one
ethyl 4-({[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}amino)piperidine-1-carboxylate
{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}[1-(1-methyl-1H-pyrazol-5-yl)propyl]amine
3-(3,5-dimethylphenyl)-1-{4-[2-(1H-imidazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(oxan-4-yl)piperazine
9-[2-(3-hydroxyphenyl)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)-2-(pyridin-3-yloxy)acetamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(dimethylamino)butanamide
1-(cyclohexylmethyl)-6-oxo-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
{imidazo[1,2-a]pyridin-3-ylmethyl}(methyl){[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}amine