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ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-(oxan-4-yl)piperidin-4-yl]acetate
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)imidazo[1,2-a]pyridine-3-carboxamide
N-{1-oxaspiro[4.5]decan-3-yl}-1H-pyrazole-4-carboxamide
2-({4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
3-{[(2-methanesulfonamidoethyl)carbamoyl]amino}-N-(2-methylpropyl)benzamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(4-phenylbutan-2-yl)piperidine
N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
4-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-oxazolidin-2-one
4-[(4-methoxy-3-methylphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-chloro-2-[(1,1-dioxo-1λ6-thiomorpholin-4-yl)methyl]phenoxy}acetic acid
2-[(2-ethyl-6-methylpyrimidin-4-yl)amino]-N-(5-fluoro-2-methylphenyl)propanamide
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)[(1-methyl-1H-indol-6-yl)methyl]amine
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(thiophen-3-ylmethyl)piperidine
1-methoxy-8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1,8-diazaspiro[4.5]decan-2-one
N-(2-hydroxyethyl)-N-methyl-2-{5-[morpholin-4-yl(phenyl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
N-[(2R,4R,6S)-2-cyclohexyl-6-(3-fluoro-2-methylphenyl)oxan-4-yl]acetamide
7-(cyclopropylmethyl)-2-(furan-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-[(2S,4R)-1-(adamantan-2-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
N-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}-3-(1H-pyrazol-1-yl)benzamide
2-amino-4-(1H-indol-5-yl)-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-[(4,5-dimethylfuran-2-yl)methyl]-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-1-ethylpiperidine-4-carboxamide
N-{1-[1-(3-fluoropyridin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-2-(thiophen-2-yl)ethan-1-one
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-[(1-methyl-1H-imidazol-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-(2,6-dimethylphenoxymethyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-{4-[1-(3-ethyl-1,2-oxazole-5-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
3-(azocan-1-yl)-N-(2,3-dihydroxypropyl)propanamide
1-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
6-methyl-5-[5-(1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(2-methylphenyl)-4-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetyl]piperazin-2-one
3-amino-1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
[1-(1H-1,3-benzodiazol-2-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
(4aS,7aR)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3S,4S)-4-methyl-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidine-3,4-diol
4-{1-butyl-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
1-[3-({3-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
6-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyridine-2-carboxamide
N-ethyl-7-[(2-fluoro-5-methoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
2-amino-3-ethyl-N-(piperidin-4-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-{4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}pentane-1,4-dione
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
6-butyl-2-{2-[(2-methylpyrrolidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
(3R,4S)-4-cyclopropyl-1-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-3-amine
methyl (2S,4S)-4-[2-(adamantan-1-ylsulfanyl)acetamido]-1-methylpyrrolidine-2-carboxylate
[(3R,4R)-1-(4,6-dimethylpyridine-3-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(4S)-3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-phenyl-1,3-oxazolidin-2-one