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5-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-3-(2-methylphenyl)pyrrolidin-3-ol
3-butanamido-4-methyl-N-(oxolan-2-ylmethyl)benzamide
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](propyl)(pyridin-3-ylmethyl)amine
1-methyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
7-methyl-2-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-phenylpiperidin-3-amine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
9-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(2-methoxyphenoxy)-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-4-carboxylic acid
1'-(4-methylpyridine-3-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-(4-{[({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]methyl}phenyl)acetamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(4-fluorophenyl)methyl]-N-methylpyrimidin-2-amine
2-(ethylsulfanyl)-5-{1-[4-(1H-pyrazol-5-yl)phenyl]-1H-imidazol-2-yl}pyrimidine
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(oxan-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N4-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[2-(7-methyl-1H-indol-3-yl)ethyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-(4-methoxypiperidin-1-yl)ethan-1-one
2-{4-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}-N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)acetamide
7-methyl-2-(naphthalen-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-[(2-methylpyridin-3-yl)oxy]-1-[3-(1H-pyrrol-1-yl)propanoyl]piperidine-4-carboxylic acid
(2R)-2-amino-3-(ethylsulfanyl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
1-(3-methoxyphenyl)-4-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)pyrrolidin-2-one
N-{[6-methyl-2-(2-methylphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-2-carboxamide
4-fluoro-3-[2-(pyridin-2-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
3-{1-[(2,6-dimethoxyphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
(1-{[1-(1-benzylpyrrolidin-3-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
2-methanesulfonamido-N-[(3R,4S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
5-chloro-2-[(3S)-3-fluoropyrrolidine-1-carbonyl]-3-phenyl-1H-indole
N-cyclohexyl-3-{[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]amino}propanamide
1-[2-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)-2-oxoethyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[2-(2-chlorophenyl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-(propan-2-yl)-4-[(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)amino]pyridine-2-carboxamide
3-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)benzoic acid
N-(1H-1,3-benzodiazol-2-yl)-5-(1-propanoylpyrrolidin-2-yl)thiophene-2-carboxamide
1-(2-hydroxyethyl)-3-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]-1-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
2-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyridine-4-carboxamide
(1S,2S)-N2-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-2,3-dihydro-1H-indene-1,2-diamine
6-(aminomethyl)-N,2-dimethyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]pyrimidin-4-amine
[2-(3-methyl-3-phenylpiperidin-1-yl)-2-oxoethyl]urea
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)pyrrolidine-3-carboxylic acid
2-{[4-(2,4-difluorophenyl)-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(2R,3R,6R)-5-(furan-3-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(piperidin-1-ylmethyl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
1-ethyl-5-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
7-(2-hydroxyethyl)-2-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
5-[1-(8-chloroquinoline-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-ethyl-1-(3-{[(4-fluorophenyl)methyl]sulfanyl}propanoyl)pyrrolidine-3-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-(2H-1,3-benzodioxole-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
2-(1-propylpiperidin-4-yl)-1-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazin-1-yl}ethan-1-one