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2-hexanoyl-N-(oxolan-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-(1-oxo-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-2-yl)methanesulfonamide
N-[1-(1-cyclopentylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxybenzamide
methyl 4-(2-amino-3-cyano-6-cyclohexyl-5-methylpyridin-4-yl)-1H-pyrazole-3-carboxylate
1-[(4-methylphenyl)methyl]-4-[2-(pyrrolidin-1-yl)butanoyl]piperazin-2-one
1-(3-chloro-4-methoxyphenyl)-5-oxo-N-[2-(1,3-thiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
1-(3-chloro-2-fluorophenyl)-3-methyl-3-[3-(1-methyl-1H-imidazol-2-yl)propyl]urea
2-(1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)-1,3-benzoxazole
8-[(2S)-2-aminopropanoyl]-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(morpholin-4-yl)propanamide
2-{2-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-(3-chloro-2-methylphenyl)-N'-ethyl-N'-(pyridin-4-ylmethyl)propanediamide
7-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-2,7-diazaspiro[4.5]decane
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(4-methylphenyl)-5-(pyridin-4-yl)pyrimidin-2-amine
(2S,3R)-2-{3-[(4-fluorophenyl)formamido]propanamido}-3-hydroxybutanamide
methyl 2-[butyl(methyl)sulfamoyl]-6-[(3-chloro-4-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(cyclopropylmethyl)-7-fluoro-3-methyl-N-propyl-1H-indole-2-carboxamide
1-(2-{1-[(3-chlorophenyl)methyl]-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl}ethyl)-1H-1,2,3,4-tetrazole
8-(cyclohex-3-en-1-ylmethyl)-3-ethyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-{4-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
6-(1-benzothiophene-2-carbonyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-{2-oxo-2-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}-1,3-thiazolidine-2,4-dione
N-[3-(1H-pyrazol-1-yl)phenyl]-3-(pyrrolidine-1-carbonyl)piperidine-1-carboxamide
N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
2-({[2-(furan-2-ylmethyl)-3-hydroxypropyl]amino}methyl)-6,8-dimethylquinolin-4-ol
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N,N-dimethylacetamide
(3S,4S)-1-(2-hydroxy-5-methylbenzoyl)piperidine-3,4-diol
2-(3-acetyl-2-fluorophenyl)-2-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}acetic acid
(3aS,6aS)-2-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{2H,4H,5H,6H-cyclopenta[c]pyrazol-2-ylmethyl}-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
2-(5-fluoropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-{4-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}cyclohex-3-ene-1-carboxamide
3-[1-(4-ethenylbenzoyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-({8-[4-(1H-pyrazol-4-yl)butanoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
1-(4-{4-chloro-2-[2-(3-hydroxypropyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
N-ethyl-N-(pyridin-4-ylmethyl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
5-phenyl-2-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}-2H-1,2,3,4-tetrazole
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(1,2,4-oxadiazol-3-ylmethyl)piperidine-4-carboxamide
1-methyl-4-({1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-yl}amino)pyrrolidin-2-one
2-{3-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-N-methylacetamide
2-[2-(5-tert-butyl-1H-1,3-benzodiazol-2-yl)phenoxy]acetamide
5-[(2R)-2-hydroxy-3-methylbutanoyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(3-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[3-(dimethylamino)phenyl]-3-[3-(1H-imidazol-2-yl)propyl]urea
3-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-methyl-1H-indole
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
3-ethyl-4-methyl-N-[2-(methylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(3-methylphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(2,3-dihydro-1H-indol-1-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one