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3-(4-fluorophenyl)-4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazin-2-one
1-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidine-3-carboxamide
4-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-acetyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]piperidine-3-carboxamide
(4aS,7aR)-1-[2-(2,3-dimethylphenoxy)acetyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(3-chloro-2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
N-[2-hydroxy-3-(pyrrolidin-1-yl)propyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-ethyl-9-(oxane-4-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
1-[2-(methylsulfanyl)ethyl]-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazine
8-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(1-{1-[2-(2-chloro-6-fluorophenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
3-(furan-2-yl)-3-[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]propanoic acid
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-N-(furan-3-ylmethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
methyl[(2-phenylphenyl)methyl](pyrazin-2-ylmethyl)amine
1,3-dimethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-{5-[1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)piperidin-3-yl]-1,2,4-oxadiazol-3-yl}pyridine
2-{4-[(6-methylpyridin-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
[5-({1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-4-yl}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
(3S,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(hydroxymethyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[4-(6-methoxypyrimidin-4-yl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
N-(5-methyl-1,2-oxazol-3-yl)-2-[2-(1H-pyrazol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(2R)-2-[(1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]propanamide
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
methyl 3-(2-methylbutanamido)-5-[(oxan-4-yl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]acetamide
2-(2,3-difluorophenoxymethyl)-N-[(5-methylpyrazin-2-yl)methyl]-1,3-oxazole-4-carboxamide
1-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
4-{4-[(2-hydroxyethyl)(methyl)amino]benzoyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
(3aS,6aR)-5-(4-methyl-1H-imidazole-2-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-(cyclopropylmethyl)-9-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-ethyl-2-(2-fluorophenyl)-5-(4-methoxypiperidine-1-carbonyl)-1H-1,3-benzodiazol-7-yl]acetamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N,N,6-trimethylpyrimidin-2-amine
(1S,5R)-6-benzyl-3-[(2-ethylpyrimidin-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-chloro-N-[(2R)-1-hydroxypropan-2-yl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
(2S,4S)-4-{[(2,6-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
1-{2-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethyl}pyrrolidin-2-one
7-methyl-3-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
1-cyclobutanecarbonyl-3-[2-(3-fluorophenyl)ethyl]piperidine
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(2-methyl-1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(4-methylphenyl)propan-2-yl]-3-(1,2-oxazinan-2-yl)propanamide
7-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one