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3-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-4-chloro-1-methyl-1H-pyrazole
2-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanamide
(2S,3S)-1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-methyl-2-(methylamino)pentan-1-one
N-[(2-methyloxolan-2-yl)methyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-({[1-(ethoxymethyl)cyclopropyl]methyl}sulfamoyl)-N-(propan-2-yl)benzamide
1-(2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
N-[5-({[3-(1H-imidazol-2-yl)propyl]carbamoyl}amino)-2-methoxyphenyl]propanamide
8-[3-(1H-pyrazol-1-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
(3aS,6aS)-2-cyclopentyl-5-[2-(dimethylamino)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-cyclopentyl-4-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-1,4-diazepane
1-benzyl-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2S,4R)-N-[(1R)-1-(4-chlorophenyl)ethyl]-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-{2-[4-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-4-(thiophen-2-ylmethyl)piperazin-2-one
3-{1-[3-(2-chlorophenyl)propanoyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
2-{4-[2-chloro-5-(trifluoromethyl)benzoyl]morpholin-3-yl}acetic acid
3-{1-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carbonyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethyl)piperazine
4-(cyclopropylmethyl)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-[(2-fluorophenyl)methyl]-N-[1-(4-methoxyphenyl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
[(1-cyclohexylpiperidin-3-yl)methyl][(2,5-dimethoxyphenyl)methyl](pyridin-3-ylmethyl)amine
2-[(5-propyl-1,2-oxazol-3-yl)formamido]-2-[2-(trifluoromethyl)phenyl]acetic acid
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N,1-dimethyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
3-methyl-4-(1-methyl-1H-pyrazol-5-yl)-1-phenyl-1H-pyrazol-5-amine
1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]but-2-yn-1-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
(2S,4R)-4-amino-1-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
2-(pyridin-2-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(dimethylamino)ethan-1-one
1-(5-methoxyfuran-2-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
6-ethyl-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-4-carboxamide
2-[2-(4-fluorophenoxy)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(phenylamino)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidine-5-carboxamide
3-[2-(3-methoxypropyl)piperidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
3-({[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]amino}methyl)piperidin-3-ol
N-[(2-amino-1,3-thiazol-4-yl)methyl]-5-{[benzyl(methyl)amino]methyl}-1,2-oxazole-3-carboxamide
8-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(3,3-diphenylpropyl)-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
9-ethyl-4-[2-(2-fluorophenyl)acetyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-ethyl-1-methyl-3-{1-[(E)-2-phenylethenesulfonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(3-methylfuran-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}benzoic acid
2-amino-4-ethyl-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,3-thiazole-5-carboxamide
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
1-{2-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazol-1-yl}propan-2-ol
1-(1,3-thiazol-4-ylmethyl)-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
8-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-8-azaspiro[4.5]decane-7,9-dione