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butyl 4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
5-{imidazo[1,2-a]pyridine-6-carbonyl}-2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
N-ethyl-7-fluoro-2-(2-methylpyrimidin-5-yl)-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
2-[1-(1-cyclopentanecarbonylpiperidine-4-carbonyl)piperidin-2-yl]pyridine
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-(4-methanesulfonylphenyl)ethan-1-one
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[2-(1H-imidazol-1-yl)ethyl]piperazine
4-[2-(2-methoxyphenyl)pyrimidin-5-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
3-(oxolan-3-yl)-5-(2-phenoxyphenyl)-1,2,4-oxadiazole
3-(2,6-dimethoxypyridin-3-yl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
2-{1-[(4-ethylphenyl)methyl]-5-[(2-oxo-1,3-oxazolidin-3-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-1,6-dimethyl-1,4-dihydroquinolin-4-one
10-methoxy-N-(1-methyl-1H-indazol-6-yl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carboxamide
N,3,4-trimethyl-5-sulfamoyl-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
N-{3-[(pyridin-3-yl)amino]propyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
2-(pyridin-2-ylsulfanyl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
4-methyl-7-{[3-(pentan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazine
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-methylpyridine-3-carboxamide
3-chloro-2-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1H-indole
N-methyl-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-2-carboxamide
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl})amine
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
(2R,6R)-4-[(2-ethyl-1,3-thiazol-4-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
methyl 3-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-{5-[4-(propan-2-yloxy)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}morpholine
N-(4,4-dimethylpentyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
2-(2,4-dichlorophenoxy)-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)acetamide
1-phenyl-3-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]pyrrolidin-2-one
(4S,4aS,8aS)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-phenyl-decahydroquinolin-4-ol
3-(2-oxo-2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethyl)imidazolidine-2,4-dione
2-methyl-3-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridine
{1-[(1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanamine
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-(4-ethenylphenyl)-2-(morpholin-4-ylmethyl)-1,4-oxazepane-4-carboxamide
9-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(furan-2-ylmethyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl](3-methylbutan-2-yl)amine
N-[(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)methyl]cyclobutanecarboxamide
(4aR,7aS)-N,N-dimethyl-4-[3-(2-methylphenyl)propanoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-methyl-5-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(3-chloro-4,5-diethoxyphenyl)methyl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
N-(3-chloro-4-methylphenyl)-2-[4-(furan-3-ylmethyl)morpholin-3-yl]acetamide
N,N-dimethyl-3-({[2-(pyridin-2-yl)ethyl]carbamoyl}methyl)morpholine-4-carboxamide
N-[(2,3-difluoro-4-methylphenyl)methyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]benzamide
5-ethyl-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1,3,4-oxadiazol-2-amine
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide