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N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]furan-2-carboxamide
6-[3-(dimethylamino)pyrrolidin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-(furan-2-ylmethyl)pyrimidin-2-amine
(4aS,7aR)-1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclopropyl-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-methyl-2-(pyrrolidin-1-yl)propyl]-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
8-{[3-(4-chlorophenyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
4-(5-methylpyridin-2-yl)-1-[6-(propan-2-yl)-1H-indole-2-carbonyl]piperidin-4-ol
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2-[(thiophen-2-ylmethyl)amino]benzamide
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-4-(5-methylfuran-2-yl)benzamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)ethan-1-one
N-(1,4-dioxan-2-ylmethyl)-3-phenoxypropanamide
1-{3-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
3-({[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-methoxy-6-methylbenzamide
N-cyclopropyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N,2-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
2-[4-(2-methoxyethoxy)phenyl]-N-methylpyridine-4-carboxamide
2-chloro-5-fluoro-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}benzamide
7-[2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzenesulfonyl]-2-oxa-7-azaspiro[4.5]decane
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
1-[(4-methylphenyl)methyl]-4-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazole
3-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazine-1-carbonyl}-5-fluorobenzonitrile
N-ethyl-5-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyrimidin-2-amine
7-(3-phenylpropyl)-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-3-(5-methylthiophene-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-phenyl-5-[(propan-2-yl)sulfamoyl]benzoic acid
N-[(2-methoxyphenyl)methyl]-N-methyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
(2S)-3-methyl-2-{4-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}butanamide
N-methyl-N-{[5-({methyl[2-(2-oxopiperidin-1-yl)ethyl]amino}methyl)furan-2-yl]methyl}methanesulfonamide
4-[1-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperidine-3-carbonyl]morpholine
3-(2-methyl-1H-indol-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
4-[2-(aminomethyl)-7-fluoro-2,3-dihydro-1-benzofuran-5-yl]pyridin-2-amine
N-[2-(4-methoxyphenyl)ethyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(4-methylphenyl)-4-[3-(trifluoromethyl)benzoyl]piperazin-2-one
2-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,8-diazaspiro[4.5]decane
N,N-dimethyl-N'-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanediamide
(2S,4S,5R)-2-ethyl-4-[(3-hydroxypropyl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
5-tert-butyl-4-({3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}methyl)furan-2-carboxamide
methyl({[1-(morpholin-4-yl)cyclohexyl]methyl}){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
5-{4-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-(3,5-dimethoxyphenyl)-3-{1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperidin-3-yl}propanamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(2,5-dioxoimidazolidin-1-yl)acetamide
1'-(3-chloro-4-methoxybenzoyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-(1-benzofuran-2-yl)pyrimidin-2-amine
9-(2-ethoxy-5-methylbenzenesulfonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
N-(1-{[1-(2-hydroxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-1H-pyrazol-5-yl)furan-2-carboxamide
(3R,4R)-1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1'-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one