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4-[4-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)piperidin-1-yl]-N-[2-(morpholin-4-yl)ethyl]benzamide
(3R,4R)-4-ethyl-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidine-3,4-diol
3-cyclohexyl-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazole
(1S,5R)-6-(3-propyl-1H-pyrazole-4-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(adamantan-1-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(4-fluorophenyl)-N-methyl-2-(piperidin-1-yl)-N-(quinolin-6-ylmethyl)acetamide
1-(4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
5-{1-[(5-chlorothiophen-2-yl)methyl]-1H-imidazol-2-yl}-2-(pyridin-2-yl)pyrimidine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-4-yl}propanamide
N-ethyl-5-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrimidin-2-amine
N-{1-[1-(1-benzylpyrrolidin-3-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
7-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]sulfonyl}-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
1-ethyl-3-methyl-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1-(4-methylphenyl)cyclopropane-1-carboxamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(quinolin-2-yl)pyrrolidin-3-yl]acetamide
N-(furan-2-ylmethyl)-1-(2-methoxyacetyl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-(3,4-dimethoxyphenyl)-1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}propan-1-one
(1S,5R)-3-methyl-6-[4-(5-methylfuran-2-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-(azepan-1-yl)-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(pyrazin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
N-[4-chloro-3-(ethylcarbamoyl)phenyl]azocane-1-carboxamide
7-(3-ethyl-1H-indole-2-carbonyl)-2,7-diazaspiro[4.5]decane
(3S,4R)-4-(2-methoxyphenyl)-1-(2-methyl-1,3-thiazole-4-carbonyl)pyrrolidine-3-carboxylic acid
5-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
3-({butyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)pyrrolidin-3-ol
2-methyl-4-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-6-(piperidin-4-yl)pyrimidine
2-({[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
7-(2-methylphenyl)-4-(3-methylpyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(1,3-dihydroxy-2-methylpropan-2-yl)-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
5-fluoro-1,3-dimethyl-2-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]-1H-indole
2-cyclopropyl-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(2-aminoethyl)-4-(2-phenoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(2H-1,3-benzodioxol-4-ylmethyl)-1-(oxan-4-ylmethyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[5-(propan-2-yl)pyrimidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(2R,3S,6R)-5-benzyl-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-3-(pyridin-3-yl)propan-1-one
6-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-N-ethylpyridine-3-carboxamide
(3S,4S)-4-(1H-imidazol-2-yl)-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
2-amino-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(propan-2-yl)pyrimidine-4-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-cyclopentyl-1H-pyrazole-3-carboxamide
1-(cyclohexylmethyl)-4-{[(3-hydroxyphenyl)methyl]amino}pyrrolidin-2-one
N-[2-hydroxy-2-(4-methoxyphenyl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
(1S,5R)-3-[4-(1H-imidazol-1-yl)butanoyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-chloro-4-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-6-methoxyphenol
4-[(2,5-difluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-2-(trifluoromethyl)benzene-1-sulfonamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-ethylpyrrolidine-3-carboxamide