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N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-1-(2-hydroxyethyl)piperidine-4-carboxamide
8-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
(3R,4R)-4-(azepan-1-yl)-1-[(3-ethoxyphenyl)methyl]piperidin-3-ol
3-(3-methoxypropyl)-1-[1-(2-methylphenyl)piperidin-4-yl]piperidine-3-carboxylic acid
(1S,5R)-6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]propan-1-one
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(thiophen-2-yl)ethyl]amine
3-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-N-(1,3-thiazol-2-yl)propanamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperazine
7-{[4-(propan-2-yl)phenyl]methyl}-2-(propane-2-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
1-(4-hydroxybutan-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(1-butyl-1H-imidazol-2-yl)-1-[3-(1H-imidazol-2-yl)benzoyl]piperidine
4-(3-hydroxy-3-methylbutyl)-N-[1-(1H-indol-2-yl)ethyl]-N-methylbenzamide
(3S,4R)-4-(hydroxymethyl)-1-{[4-(2-methylphenyl)phenyl]methyl}piperidin-3-ol
N-(5-methyl-1,2-oxazol-3-yl)-2-(oxolane-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
8-{2-[5-oxo-2-(thiophen-2-yl)cyclopent-1-en-1-yl]acetyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
8-(5-chloro-2-hydroxybenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-5-(4-methoxyphenyl)furan-2-carboxamide
5-[2-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2,3-dihydro-1H-isoindol-2-yl)-1-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]ethan-1-one
N,N-dimethyl-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrazin-2-amine
methyl 5-oxo-5-{3-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}pentanoate
9-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
(2S,4S)-4-amino-N-methyl-1-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]pyrrolidine-2-carboxamide
3-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]naphthalene-2-sulfonamide
1-(2-methoxyethyl)-3-(propan-2-yl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(methylsulfanyl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}pyrimidine-5-carboxamide
5-({[2-amino-6-(propan-2-yl)pyrimidin-4-yl]amino}methyl)-1,2,4-oxadiazole-3-carboxamide
({4-cyclopropyl-5-[1-(trimethylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
2-{2-[2-(hydroxymethyl)phenyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
2-methyl-5-[(3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2-oxazol-5-yl)methoxy]-1,3-benzothiazole
2-[(4-fluoro-3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-(3-chlorophenoxy)-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]ethan-1-one
(3aR,6aR)-2-benzyl-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
[(2S,4R)-4-(dimethylamino)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidin-2-yl]methanol
ethyl 5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}adamantan-1-yl acetate
N,N-dimethyl-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
3-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}morpholine
2-hydroxy-4-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]pentanamide
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-2-amine
3-(2-fluoro-4-methoxyphenyl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
4-[(5-methylfuran-2-yl)methyl]-3-{2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}piperazin-2-one
2-[5-({5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}methyl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
6-[1-(3-benzyl-1H-1,2,4-triazol-5-yl)ethoxy]-4-methyl-2H-chromen-2-one
N-methyl-N-{1-[2-(pyridin-4-yl)-1H-imidazol-1-yl]propan-2-yl}aniline