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1-(2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]amine
3-[2-(6-hydroxy-1,4-oxazepan-4-yl)-2-oxoethyl]-3,4-dihydroquinazolin-4-one
5-propyl-1'-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-fluoro-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylquinoline-2-carboxamide
5-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-2,3-dimethylbenzene-1-sulfonamide
N-cyclohexyl-5-(1-{[ethyl(methyl)sulfamoyl]amino}ethyl)-N,4-dimethylpyrimidin-2-amine
3-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-methylpyrrolidine-2-carboxamide
N-methyl-N-(1-methylpiperidin-4-yl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-ethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{[1-(methoxymethyl)cyclopropyl]methyl}acetamide
3-(2-methoxyethyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
1-[2-({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)ethyl]imidazolidin-2-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
3-chloro-5-[1-cyclohexyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
7-(2-methyl-1-benzofuran-5-carbonyl)-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-(carbamoylmethoxy)-N-(2-methoxyethyl)-N-(oxolan-2-ylmethyl)benzamide
2-(1-methyl-1H-pyrrol-2-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-oxoacetamide
2-{4-[4-(1,3-benzothiazol-2-yl)-1,4-diazepane-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
2-(benzyloxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
6-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methyl-1,3-benzoxazole
8-[(4-methylphenyl)methanesulfonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-(furan-3-carbonyl)-N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[(2-chlorophenyl)methyl]-5-(piperidin-4-yl)-3-(pyridin-3-ylmethyl)imidazolidine-2,4-dione
4-methyl-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
N-(2-hydroxy-3-methoxypropyl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
(1R,5R)-3-cyclobutanecarbonyl-6-[(2,4-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(2R,3R)-3-(piperidin-1-yl)-1'-(pyridin-4-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-benzyl-1-[(1-ethylpyrrolidin-3-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopropyl-4-methoxy-3-[(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)oxy]benzamide
2-methyl-1-{2-oxo-2-[3-(propoxymethyl)pyrrolidin-1-yl]ethyl}-1,4-dihydroquinolin-4-one
1-{4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(1,3-thiazol-4-yl)ethan-1-one
1-(2H-1,3-benzodioxol-4-ylmethyl)-4-[(3-fluorophenyl)methyl]piperazine
4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[3-(2-methoxyphenoxy)azetidin-1-yl]isoquinoline
N-methyl-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-(quinolin-2-ylmethyl)acetamide
2-(3-chlorophenyl)-2-hydroxy-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}pyrimidin-2-amine
6-(pyrrolidin-1-ylmethyl)-4-(1,3-thiazol-4-ylmethyl)-1,4-oxazepan-6-ol
(3aS,6aS)-2-(cyclopropylmethyl)-5-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-methyl-N-[2-(3-methylpiperidin-1-yl)ethyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
1-(2-{[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}ethyl)imidazolidin-2-one
2-[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]ethan-1-amine
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1,4-dihydropyridine-3-carboxamide
(4aS,8aR)-6-(6-methoxypyrimidin-4-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
9-(5-chloro-2-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{2-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-(pyridin-4-yl)ethyl}morpholine
2-methylpropyl 4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
8-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one