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dimethyl(2-{2-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
2-(cyclohexylmethyl)-4-(thiophene-3-carbonyl)morpholine
3-{2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamido}propanamide
2-(6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-3-yl)acetic acid
1-({5-[(4-methoxy-3-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
4-(benzyloxy)-1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
2-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
6-(2-phenyl-1H-imidazol-1-yl)pyridin-2-amine
3-({[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-4-yl]oxy}methyl)pyridine
3-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}oxy)-N-(2-phenylethyl)benzamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-4-carboxamide
1-[2-(4-ethoxypiperidin-1-yl)-2-oxoethyl]-3-methyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
9-(2-hydroxy-3-methylbutanoyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-[2-(dimethylamino)benzoyl]-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidine-1-carbonyl]pyridin-3-ol
N-[2-(ethylsulfanyl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
6-methoxy-2-oxo-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl 6-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]pyrimidine-4-carboxylate
2-cyclopropyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
1-{1-[6-(4-hydroxypiperidin-1-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-3-(pyrazin-2-yl)propanamide
2-amino-1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]propanamide
N-[2-(1H-pyrazol-4-yl)ethyl]-2H-1,3-benzodioxole-5-carboxamide
4-(5-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}-1H-pyrazol-3-yl)phenol
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
6-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-methyl-N-[1-(thiophen-2-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
(2S,4R)-4-(cyclooctylamino)-N-ethyl-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
9-(1,4-dithiepan-6-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)benzamide
4-chloro-1,5-dimethyl-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-3-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
9-[(3-chloro-4-fluorophenyl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-6-(propan-2-yloxy)pyrimidin-2-amine
2-methyl-5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]pyrimidin-4-ol
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-[2,5-dioxo-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-(oxan-2-ylmethyl)acetamide
2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(piperidin-1-yl)acetamide
1-[(3-chlorophenyl)methyl]-N-[3-(propan-2-yloxy)propyl]-1H-1,2,3-triazole-4-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(naphthalen-2-yloxy)propanamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-(2-ethyl-1H-1,3-benzodiazol-6-yl)urea
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[(5-methoxy-1H-indol-2-yl)methyl]acetamide
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
4-methyl-N-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1,2,3,6-tetrahydropyridine-1-carboxamide
(3S,4R)-4-(hydroxymethyl)-1-[3-(pyrrolidine-1-sulfonyl)thiophene-2-carbonyl]piperidin-3-ol
4-(4-chlorobenzenesulfonyl)piperazine-2-carboxylic acid
6-methoxy-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2,3-dihydro-1H-indene-5-carboxamide