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N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-4-(trifluoromethyl)benzamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-cyclopropyl-9-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
(3S,9aR)-3-benzyl-8-(3-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-cyclopropyl-2-fluoro-N-[(2-methoxyphenyl)methyl]-5-sulfamoylbenzamide
N-(3-methylphenyl)-3-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-4-yl}propanamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-(2-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)acetic acid
(1R,5R)-6-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[2-(pyrazin-2-yl)ethyl]-1-benzofuran-5-carboxamide
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-ylmethyl]-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-(quinoxalin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-{1-[(6-fluoroquinolin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
2-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]-1-(piperazin-1-yl)ethan-1-one
(2S,4S)-4-acetamido-N-ethyl-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}pyrrolidine-2-carboxamide
2-[(2,6-dichlorophenyl)methyl]-5-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
N-cyclopropyl-N-(1-{1-[(2E)-4-methylpent-2-en-1-yl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
(3S,4R)-3-benzyl-1-[(5-fluoro-2-methoxyphenyl)methyl]-4-methylpiperidin-4-ol
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N-(3,5-dimethoxyphenyl)-3-{1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-3-yl}propanamide
5-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-5,6-dihydrophenanthridin-6-one
3-{[(3R,4S)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-(oxane-4-carbonyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2-methyl-1-benzofuran-5-carboxamide
N-(1-propylpiperidin-3-yl)-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-(furan-2-ylmethyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-(3-hydroxypropyl)-8-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-({4-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}methyl)azetidin-3-ol
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-2-methoxy-N-(pyridin-3-ylmethyl)benzamide
{[5-(3-chlorophenyl)furan-2-yl]methyl}(methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
2-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
1-(1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-(propan-2-yl)piperidine-4-carboxamide
N'-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N'-[2-(dimethylamino)ethyl]-N,N-dimethylbutanediamide
2-[1-(1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-methylpiperidine
9-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[4-(4-fluorophenoxy)piperidine-1-carbonyl]-5-methyl-4,5,6,7-tetrahydro-2H-indazole
1-methyl-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(3R,4S)-1-(2-chloro-6-methylbenzenesulfonyl)-4-(dimethylamino)piperidin-3-yl]propanoic acid
5-{[3-(1-benzofuran-2-yl)-1H-pyrazol-1-yl]methyl}-3-(cyclopropylmethyl)-1,2,4-oxadiazole
1-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-2-(pyridin-3-yl)ethane-1,2-dione
N-[(3R,4S)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)-N-methylpropanamide
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-2-(1-methyl-1H-imidazol-2-yl)benzamide
10-methoxy-5-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-({[4-(methylsulfanyl)phenyl]methyl}({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})amino)ethan-1-ol
2-[9-(1-methylpiperidine-3-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
3-(2-methoxyethyl)-5-({5-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
1-(4-amino-5-methylpyrimidin-2-yl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid