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N-{[2-(azepan-1-yl)-7-fluoroquinolin-3-yl]methyl}-N-(2-methoxyethyl)acetamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(1,2-oxazolidin-2-yl)-N-(oxolan-2-ylmethyl)propanamide
(1R,2S)-N-tert-butyl-2-(4-butyl-3-oxopiperazine-1-carbonyl)cyclohexane-1-carboxamide
3-(2-methylpropyl)-N-[3-(pyridin-2-yl)propyl]-1,2-oxazole-5-carboxamide
2-(2-hydroxyethyl)-N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-3-oxopiperazine-1-carboxamide
1-(2-methoxyethyl)-3-methyl-8-[(5-methylthiophen-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3S,4R)-4-methoxyoxolan-3-yl]-3-(2-methoxyphenyl)benzamide
1-[2-(2-chlorophenyl)ethyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-[2-(pyrrolidin-1-yl)propyl]-1,2-oxazole-3-carboxamide
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
2-amino-4-(6-methoxy-1-methyl-1H-indol-3-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
3-(3-hydroxy-3-methylbutyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}benzamide
6-{1-ethyl-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}-2-methyl-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
3-{1-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
(4aR,7aS)-N,N-dimethyl-4-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-{4-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
1-benzyl-4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-1,4-diazepan-6-ol
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]pyridine-4-carboxamide
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-2,3,6-trimethylquinoline-4-carboxamide
(1R,5S,8R)-3-(1H-1,3-benzodiazole-2-carbonyl)-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
1-tert-butyl-N-[3-(2-methoxyphenoxy)propyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
1-(4-benzylpiperazin-1-yl)-3-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]propan-1-one
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(5-methylthiophen-2-yl)methyl]piperidine
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-[4-(6-ethyl-4-methylquinolin-2-yl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
5-methyl-N2-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrimidine-2,4-diamine
3-{2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
N-[2-({cyclopropyl[(2-ethoxyphenyl)methyl]amino}methyl)quinolin-6-yl]acetamide
N-cyclopentyl-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,1,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-phenyl-5-({2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1H-1,2,3,4-tetrazole
N-(adamantan-1-ylmethyl)-5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
6-[(3S)-3-hydroxy-3-phenylpropyl]-5,6-dihydro-1,6-naphthyridin-5-one
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[(3,5-dimethoxyphenyl)methyl]propanamide
4-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-4-oxobutane-1-sulfonamide
3-methyl-9-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-3,9-diazaspiro[5.6]dodecane
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-3-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}urea
N-(1-benzylpiperidin-3-yl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]benzamide
N-cyclopropyl-3-{5-[2-(thiophen-2-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-benzyl-5-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole
(2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)urea
(1S,5R)-6-benzyl-3-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(3-{[1-(3,4-dimethoxybenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
1-[cyclohexyl(methyl)amino]-3-[2-(1,2-oxazinan-2-ylmethyl)phenoxy]propan-2-ol
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(2-methylphenoxy)azetidin-1-yl]propan-1-one
4-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methylpyrimidine