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1-(2-aminoethyl)-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
6-(2-aminoethyl)-N-[(2,5-dimethylphenyl)methyl]-2-methylpyrimidin-4-amine
N-[2-(1H-imidazol-4-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-(1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)propan-1-one
N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-4-(4H-1,2,4-triazol-4-yl)benzamide
methyl 5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-5-oxopentanoate
methyl 2-[({1-[(3,4-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]acetate
2-[2-(3-methoxypyrrolidin-1-yl)-2-oxoethyl]-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl](methyl){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
(2S,4R)-N-methyl-4-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]-1-propylpyrrolidine-2-carboxamide
4-methoxy-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
1-[5-({[2-(2-fluorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-methylpyrazine
3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(thiolan-3-yl)benzamide
dimethyl({4-methyl-5-[1-(thiophene-2-sulfonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-(3-methylpyridin-4-yl)-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-diazepane
N-cyclohexyl-8-methoxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-N'-(2,4,6-trimethylphenyl)butanediamide
2-ethoxy-5-{2-[methyl(pyridin-2-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
4-ethyl-3-(piperidin-4-yl)-1-(pyrimidin-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(4-fluorophenyl)morpholin-4-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2-(5-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
N-(furan-2-ylmethyl)-1-methyl-N-(prop-2-en-1-yl)-1H-pyrrole-2-carboxamide
4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamido]-N-phenylpiperidine-1-carboxamide
2-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]-4-(methylsulfanyl)butanoic acid
methyl 5-(4-sulfamoylbenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
5,8-dimethoxy-4-methyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]quinoline
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-[(4-{7-methyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}phenyl)sulfanyl]ethan-1-ol
2-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}-5-methoxyphenol
1-({4-methyl-5-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
9-[(2-methyl-1,3-oxazol-4-yl)methyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)(oxolan-3-ylmethyl)amine
3-(diphenylmethyl)-4-(3-methoxyphenyl)-4H-1,2,4-triazole
4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylbenzamide
2-methoxy-2-phenyl-N-{1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
(4aR,8aR)-7-[4-(dimethylamino)benzoyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
(2S)-N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
3-[2-(3,4-difluorophenyl)ethyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
1-[2-({[(3-ethyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N3-cyclooctyl-N5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-4-oxobutanamide
4-(4-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}phenyl)phenol
[1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl](phenyl)methanol
N-({1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)pyrazine-2-carboxamide
1-(oxolan-2-ylmethyl)-4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazole
3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
(4aS,7aR)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione