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(2S,4R)-4-amino-N,N-diethyl-1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]pyrrolidine-2-carboxamide
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-3-(4-methylpiperazin-1-yl)propan-1-one
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
4-({5-[1-(3-cyclopentylpropyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-tert-butyl-1-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}urea
[2-(2-methyl-1H-indol-1-yl)ethyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
5-[2-(benzylamino)ethyl]-1-[3-(methylsulfanyl)propyl]pyrrolidin-2-one
dimethyl[(3-{[8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenyl)methyl]amine
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-[(3-methylphenyl)sulfanyl]piperidine
2-{5-[2-(1,3-benzothiazol-2-yl)ethyl]-3-cyclopropyl-1H-1,2,4-triazol-1-yl}acetic acid
2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-6-(pyrrolidine-1-carbonyl)pyrazine
N-(5-{pyrazolo[1,5-a]pyridin-7-yl}pyridin-2-yl)acetamide
2-(2-hydroxyethyl)-9-[(4-methoxynaphthalen-1-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3,5,7-trimethyl-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}-1H-indole
2-amino-N-cyclohexyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-fluoro-4-methylbenzenesulfonyl)-2-(3-methoxypropyl)piperidine
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-3-ylsulfanyl)acetamide
6-methyl-3-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
2-{9-[(3,4-dimethoxyphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-(2-methylphenyl)-3-phenylpropanamide
1-[5-(3-acetylphenoxymethyl)-1H-pyrazole-3-carbonyl]-N-methylpyrrolidine-3-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(cyclobutylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-chloro-4-fluoro-N-(1-methyl-2-oxopyrrolidin-3-yl)-1-benzothiophene-2-carboxamide
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(2-methoxyethyl)methylamine
6-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-(3-hydroxyquinoxalin-2-yl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]propanamide
1-(2-methoxy-4-{[(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
7-cyclopropanecarbonyl-N-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-(1H-imidazol-2-ylmethyl)-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(dimethylamino)ethyl]-2-(2,4-dioxo-1,3-diazinan-1-yl)-N-methylbenzamide
3-(1-methyl-1H-pyrazol-4-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-cyclopropanecarbonyl-8-{[4-(propan-2-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 5-[3-(1,2-oxazinan-2-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
5-(2-chloro-6-methoxyphenyl)-4-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
(2E)-1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-phenylprop-2-en-1-one
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-4-hydroxypiperidine-4-carboxylic acid
5-(morpholine-4-carbonyl)-2-(3-phenylpropyl)-1,3-benzoxazole
1-(2-ethylphenyl)-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[2-(morpholin-4-yl)propyl]acetamide
N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-4-(piperidin-3-yl)benzamide
3-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-2-methyl-6H,7H-pyrazolo[1,5-d][1,2,4]triazin-7-one
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N3-(4-fluorophenyl)-N5-[2-(1H-indol-3-yl)ethyl]piperidine-3,5-dicarboxamide
2-{4-[1-(morpholin-4-yl)ethyl]phenyl}-N-propylbenzamide
N-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
4-(3,4-difluorobenzoyl)-1-{imidazo[1,2-a]pyridine-6-carbonyl}piperidine
N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-cyclopentyl-3-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]propanamide
N-[3-(4-{[1-(1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-3-(trifluoromethyl)benzamide