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6-(benzyloxy)-4-[(2,3-difluorophenyl)methyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-[4-(1H-pyrazole-4-carbonyl)-1,4-diazepan-1-yl]-1,3-benzothiazole
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(5-fluoro-1H-indol-2-yl)methyl]methylamine
(1S,5R)-1,3,3-trimethyl-6-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-6-azabicyclo[3.2.1]octane
5-fluoro-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-indole-2-carboxamide
2-(1-methyl-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-yl)ethan-1-ol
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methyl-N-(2-methylprop-2-en-1-yl)pyridin-2-amine
(4aS,7aR)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-ethyl-3-methyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
(3aR,6aR)-2-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-[(3,4-difluorophenyl)methyl]-8-(2-hydroxyacetyl)-2,8-diazaspiro[4.5]decan-3-one
3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}urea
2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
1-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}-2-(pyridin-2-yl)ethan-1-one
N'-cyclohexyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-N'-methylbutanediamide
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]propanamide
4-[4-(5-fluoro-2-methoxybenzoyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
6-(2-chlorophenyl)-N-[(2S)-1-methoxypropan-2-yl]-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(2-methyl-1H-imidazol-1-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-{[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,5-dimethyl-1H-indazole
7-fluoro-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}quinazolin-4-amine
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-6-(piperidin-4-yl)pyrimidin-4-amine
2-methyl-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}thieno[2,3-d]pyrimidin-4-amine
1-[(4-chlorophenyl)methyl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-(methanesulfonylmethyl)-1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazole
3-(benzylsulfanyl)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
2-[4-(2,6-dimethoxypyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-4-(1H-pyrazol-1-yl)butan-2-ol
2-fluoro-N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenol
3-[3-(1H-1,2,4-triazol-1-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-chloro-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(quinoline-3-carbonyl)pyrrolidine-2-carboxamide
4-[3-(furan-2-yl)-1H-pyrazol-5-yl]-1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidine
1-(2-{4-[(3-ethoxy-2-hydroxyphenyl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
N-(4-methoxyphenyl)-1-[4-(trifluoromethyl)benzoyl]piperidin-3-amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-(3-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
5-chloro-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)thiophene-2-carboxamide
3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-5,6,7,8-tetrahydroquinoline
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-(2-fluorophenyl)ethyl]benzamide
1,3-dimethyl-5-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
[(2S,6S)-4-{[4-(methylsulfanyl)phenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-[(3R,4S)-1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-(1-cyclopentylpiperidine-3-carbonyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
3-{2-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}-2,3-dihydro-1λ6-thiophene-1,1-dione
6-ethyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-oxo-1,2-dihydropyridine-4-carboxamide