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7-(3,6-dimethylpyrazin-2-yl)-4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-N'-[2-(methylsulfanyl)phenyl]butanediamide
4-{4-methyl-3-[2-(1-phenylethyl)-1H-imidazol-1-yl]phenyl}-4H-1,2,4-triazole
1,3-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}pyrazin-2-ol
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-1-carboxamide
2-(4-chlorophenyl)-4-[4-(piperidine-1-carbonyl)pyridin-2-yl]morpholine
(oxolan-2-ylmethyl)(1,3-thiazol-2-ylmethyl)(thiophen-3-ylmethyl)amine
methyl 4-(3-{[4-(3-fluorophenyl)phenyl]carbamoyl}piperidin-1-yl)-4-oxobutanoate
(2S,4S)-1-(adamantan-2-yl)-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N-(3-chloro-4-fluorophenyl)-3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]propanamide
[4-methyl-5-(1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methanol
3-[2-(2-fluorophenyl)ethyl]-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
6-{4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-1-yl}pyridine-3-carbonitrile
6-[3-(3,4-dimethoxyphenyl)propanoyl]-N-phenyl-6-azaspiro[2.5]octane-1-carboxamide
8-(4-carboxypyridin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(4-methylphenyl)-4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}pyrrolidin-2-one
N-({2-[3-(2,5-dimethylfuran-3-amido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-(propan-2-yl)oxane-4-carboxamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(1H-imidazole-2-carbonyl)piperidine
5-{cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
2-{[1-(3-acetamidophenyl)-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
6-methyl-N-[1-(oxan-4-yl)piperidin-4-yl]-2-propylpyrimidin-4-amine
1-{7-[(4-benzylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}ethan-1-one
N-(3,4-difluorophenyl)-6-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(4,6-dimethylpyrimidin-2-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidin-4-amine
2-{4-[(3,5-dimethylphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-(oxan-3-ylmethyl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-[methyl({4-methyl-5-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
N-(2-{[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]amino}ethyl)pyridine-3-carboxamide
2-{4-[3-(1-methoxyethyl)phenyl]-1H-pyrazol-5-yl}pyridine
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-{[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]sulfanyl}acetamide
9-(3-fluoro-4-methylbenzoyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-1-[(2,2-difluoro-2H-1,3-benzodioxol-4-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
3-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-1-[2-(2-methoxyphenyl)ethyl]urea
3-hydroxy-3-({[3-(1H-indazol-1-yl)propyl]amino}methyl)-1-methylpiperidin-2-one
N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(pyridin-2-ylsulfanyl)acetamide
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl})amine
ethyl 1-(1H-imidazol-4-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-(2-{2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)acetamide
4-chloro-N-[1-(cyclohex-1-en-1-yl)ethyl]-1-methyl-1H-pyrazole-3-carboxamide
5-methyl-3-(2-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-2-oxoethyl)-2,3-dihydro-1H-indol-2-one
3-(3-hydroxyquinoxalin-2-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]propan-1-one
2-(2,3-difluorophenoxymethyl)-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
4-{1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}pyridine
2-{4-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
2-methoxy-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
4-(4-methoxy-2,5-dimethylphenyl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-1,2,3-triazole
5-[6-amino-5-cyano-4-(furan-2-yl)pyridin-2-yl]thiophene-3-carboxylic acid
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine