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2-amino-4-methyl-N-(5-oxo-1-phenylpyrrolidin-3-yl)-1,3-benzothiazole-6-carboxamide
5-{3-[(3,4-dimethoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-4-methyl-1,3-oxazole
1-{3-[(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)methyl]phenyl}ethan-1-one
N-(butan-2-yl)-3-[(4-fluorophenyl)formamido]-N-[(3-methylthiophen-2-yl)methyl]propanamide
N,N-diethyl-1-{[4-(quinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-3-carboxamide
N-[2-(2-fluorophenyl)-1-{1-[(2E)-3-(pyridin-4-yl)prop-2-enoyl]piperidin-4-yl}ethyl]-N-methylthiophene-2-carboxamide
4-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)morpholine
4-(4H-1,2,4-triazol-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]benzamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}pyrazine-2-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-(3-fluorophenoxymethyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidine
N-(1-methyl-1H-1,2,3-triazol-4-yl)-5-[1-(2-methylpropyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-methyl-1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidine-3-carboxamide
1,3-dimethyl-5-({[4-(pyridin-3-yl)pyrimidin-2-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
8-(1,3-benzoxazol-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-tert-butyl-2-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenoxy)acetamide
4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}propanamide
(2S,4R)-4-[(adamantan-2-yl)amino]-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
(3S,5R)-1-[(3-hydroxyphenyl)methyl]-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(3,4-difluorobenzoyl)pyrrolidin-3-yl]methanol
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
7-(1,3-benzothiazol-2-yl)-4-[(4-fluorophenyl)methyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[2-(furan-2-yl)pyrimidin-5-yl]-7-methyl-1H-1,3-benzodiazole
methyl 3-[(3S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
1-{2-[(5-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}azepane
N-(1-benzothiophen-5-ylmethyl)-2-fluoro-5-sulfamoylbenzamide
1-(oxan-4-yl)-4-(3-phenylbutyl)piperazine
[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)(quinolin-3-ylmethyl)amine
1-[(2-fluorophenyl)methyl]-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)piperidin-2-one
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
7-propyl-2-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
[(2S)-1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
(1R)-2-{3-[3-(3,6-dimethylpyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}-1-phenylethan-1-ol
9-(3,4-dimethylbenzoyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-[(1-methyl-1H-indol-6-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(2,4-difluorophenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-ol
6-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-3-carboxylic acid
(2R,3R,6R)-5-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
6-fluoro-2-[({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)methyl]quinolin-4-ol
3-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}-1-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}urea
3-methoxy-1-{2-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]acetamide
4-{3-phenyl-5-[4-(propan-2-yl)piperazine-1-carbonyl]benzenesulfonyl}thiomorpholine
5-fluoro-N-[3-(1H-imidazol-1-yl)propyl]-4-(pyrrolidin-1-yl)pyrimidin-2-amine
N-(1-{1-[1-(ethylcarbamoyl)ethyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide