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3-chloro-N-cyclopentyl-4-{[1-(thiophen-3-ylmethyl)piperidin-4-yl]oxy}benzamide
1-[(2,6-difluorophenyl)methyl]-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(3-methoxypropyl)-9-[2-(4-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(3,5-dimethylphenyl)-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperazin-2-one
N-[(5-methylpyrazin-2-yl)methyl]-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1-methyl-1,4-dihydroquinolin-4-one
methyl 2-{3-[(2-methoxyethyl)carbamoyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}acetate
2-(1-methyl-1H-imidazol-2-yl)-1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
3-[(dimethylamino)methyl]-1-{[2-(propylamino)pyrimidin-5-yl]methyl}pyrrolidin-3-ol
2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-N-(propan-2-yl)aniline
2-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,3-thiazole
6-(4-fluorophenyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-N-(2-methylpropyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(6-chloroquinolin-2-yl)-4-hydroxypiperidine-4-carboxylic acid
ethyl 6-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}pyrazolo[1,5-a]pyrimidine-3-carboxylate
3-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1H-pyrazol-5-amine
2-(2H-1,2,3-benzotriazol-2-yl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
N-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}[(2-methylphenyl)methyl]amine
3-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)benzoic acid
4-[4-(pyridin-3-yl)piperazin-1-yl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
3-(2,5-dimethylbenzoyl)-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(4-fluorophenyl)-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-4-ol
N,1-dimethyl-N-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidin-3-amine
3-(5-methylfuran-2-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-3-(2-oxopyrrolidin-1-yl)propanamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)propanamide
5-{[benzyl(methyl)amino]methyl}-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-1,2-oxazole-3-carboxamide
2-(2,2-diphenylethyl)-4-(3-methyl-1H-pyrazole-5-carbonyl)morpholine
methyl 3-[ethyl({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})carbamoyl]propanoate
3-(azepan-1-yl)-1-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]propan-1-one
2-methoxy-2-methyl-N-[(3R,4S)-4-(propan-2-yl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]propanamide
1-(piperidin-3-yl)-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
[(2S)-1-[3-(thiomorpholine-4-carbonyl)benzenesulfonyl]pyrrolidin-2-yl]methanol
(3S,4S)-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-(1H-1,2,4-triazol-3-ylsulfanyl)ethan-1-one
N-{2-[4-(methylsulfanyl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-4,4,4-trifluorobutan-1-one
[3-(cyclopropylmethyl)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-3-yl]methanol
1-[5-(2-methylbenzoyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(3-methoxypropanoyl)pyrrolidin-3-yl]-1,3-dimethyl-1H-pyrazole-4-carboxamide
(3S,5R)-N5-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-N3,N3-dimethylpiperidine-3,5-dicarboxamide
2-(3-hydroxyadamantan-1-yl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]acetamide
N-[3-(1H-pyrazol-1-yl)phenyl]-1H-indazole-3-carboxamide
6-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]pyridin-3-ol
1-(2,3-dihydro-1H-inden-2-yl)-4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]urea
4-(4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-1,3-thiazol-2-amine
2-phenyl-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]acetic acid
4-[(2-methylpyridin-3-yl)oxy]-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid