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N'-cycloheptyl-N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)butanediamide
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[(1-ethylpyrrolidin-2-yl)methyl]piperidine-3-carboxamide
ethyl 3-(2-methoxyethyl)-1-{[4-(2-oxoimidazolidin-1-yl)phenyl]methyl}piperidine-3-carboxylate
3-[(3S,4S)-1-ethyl-4-methoxypyrrolidin-3-yl]-1-[2-(3-methylphenoxy)phenyl]urea
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
8-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-methyl-7-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
N,N-diethyl-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
5-[1-(1-benzothiophene-5-carbonyl)pyrrolidin-2-yl]-3-methyl-1,2-oxazole
4-(2-methylphenoxy)-1-[(2S)-piperidine-2-carbonyl]piperidine-4-carboxylic acid
1-[4-(4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
2-methoxy-5-({3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}methyl)pyrimidine
{[2-(1H-imidazol-1-yl)phenyl]methyl}(4,4,4-trifluorobutan-2-yl)amine
2-{1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
2-(2-hydroxyethyl)-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-hydroxy-3-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)-1-[(3-methoxyphenyl)methyl]piperidin-2-one
1-[(2-phenylpyrimidin-5-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
N-[(2-chloro-4-fluorophenyl)methyl]-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
7-(3-chlorophenyl)-4-(furan-3-carbonyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-(1-benzofuran-5-ylmethyl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
(5S,9aS,9bS)-2-cyclopentyl-5-(1-phenyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[3-(4-fluorophenyl)phenyl]-1-(3-methoxypropanoyl)piperidine-3-carboxamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[3-(propan-2-yloxy)propyl]amino}methyl)phenoxy]propan-2-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)acetamide
2-(1,3-benzoxazol-2-ylsulfanyl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butan-1-one
2-({5-[1-(2-methyl-1H-1,3-benzodiazol-6-yl)-1H-imidazol-2-yl]pyrimidin-2-yl}amino)acetic acid
(3S,4R)-4-(3-methoxyphenyl)-1-(1,2-thiazole-5-carbonyl)pyrrolidine-3-carboxylic acid
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
(4aR,7aS)-1-methanesulfonyl-4-(3-phenylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl[1-(pyridin-3-yl)ethyl]{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
1-benzyl-8-(butan-2-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(furan-2-ylmethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-(1H-imidazol-1-yl)ethan-1-one
7-(cyclopropylmethyl)-2-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
1-(5-methyl-1,2-oxazole-3-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
7-cyclobutanecarbonyl-N,N-dimethyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-(3-chlorophenyl)-N-methyl-N-(2-methylpropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(4-chloro-2-fluorophenyl)-2-{[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]amino}acetamide
N-[2-(cyclohexylsulfanyl)ethyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
(1S,5R)-3-[(2-fluoro-4-methoxyphenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
1-ethyl-5-methyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-4-carboxamide
(3aR,5R,6S,7aS)-2-(1H-indol-7-ylmethyl)-octahydro-1H-isoindole-5,6-diol
N-cyclopentyl-N-({4-[(3-fluorophenyl)methoxy]-3,5-dimethoxyphenyl}methyl)-2,2-dimethyloxane-4-carboxamide
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(3-hydroxyphenyl)-N-[1-(pyridin-4-yl)propyl]acetamide
9-(5-methoxy-1H-indole-2-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
2-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethan-1-ol
3-(3-chlorophenyl)-5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole