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1-(1H-indol-7-ylmethyl)-4-(oxan-4-yl)-1,4-diazepan-6-ol
(1S,5R)-6-(dimethyl-1,3-thiazole-5-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 4-(4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)benzoate
methyl 6-{[benzyl(ethyl)amino]methyl}-3-cyclopropaneamidothieno[2,3-b]pyridine-2-carboxylate
5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
N-(cyclopropylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
2-{1-methyl-4-[1-(4-methylphenyl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{[6-(4-fluorophenyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}propanamide
3-[4-(2-methoxyethyl)piperazin-1-yl]-5-(2-methylphenyl)-1,2,4-triazine
(1S,4S)-2-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}-2-azabicyclo[2.2.1]heptane
1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-4-(3-methylpyridin-4-yl)piperazine
(4aS,7aR)-1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4S)-N-cyclopentyl-4-hydroxy-3,3,4-trimethylpiperidine-1-carboxamide
1-cyclopentanecarbonyl-3-[2-(3-methoxyphenyl)ethyl]piperidine
5-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]quinoxaline
N-ethyl-2-[4-(1H-imidazol-2-ylmethyl)piperazin-1-yl]acetamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
4-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-6-(propan-2-yl)pyrimidin-2-amine
2-[3-(difluoromethyl)-5-methyl-1H-pyrazol-1-yl]-N-ethyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
4-(dimethylamino)-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}benzamide
1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-1,2,3,4-tetrahydroquinolin-2-one
N-[(3-fluorophenyl)methyl]-2-methanesulfonamido-N-[(4-methoxyphenyl)methyl]propanamide
7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(2-{2-[1-(3-chloropyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2-{1-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-1H-1,2,3-triazol-4-yl}benzoic acid
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl){[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
5-(1H-pyrazol-1-ylmethyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}furan-2-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
2-methoxy-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-sulfamoylbenzamide
4-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-amine
3-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-(2,6-dimethoxypyridin-3-yl)urea
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-1-(pyridin-2-ylmethyl)piperidin-4-amine
(4aR,7aS)-1-(2-hydroxyethyl)-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(benzylsulfamoyl)({[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl})amine
6-[(3,5-dimethoxyphenyl)methoxy]-4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-1-(propan-2-yl)-1,4-diazepan-2-one
7-(2-benzyl-1,3-thiazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methylphenyl)methyl]piperidine
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-({4-[2-(trifluoromethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
1-(2-methoxyethyl)-8-[(5-methylthiophen-2-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1R,3R)-3-aminocyclopentyl]-9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
4-methanesulfonyl-N-[2-methyl-3-(pyrrolidin-1-yl)phenyl]piperazine-1-carboxamide
2-[(1R,3S,3aS,6aR)-1-(hydroxymethyl)-5-methyl-3-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
1-(benzylcarbamoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-[(4-methoxy-3-methylphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-[(2-methoxyphenyl)methyl]acetamide
1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4-(pyridin-4-yl)piperazine