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3-[(4-methoxyphenyl)methyl]-1-methyl-8-{[3-(2-methylphenyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperidine-4-carboxylate
1-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2-phenylethane-1,2-dione
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-1-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1H-1,2,3-triazole
2-({4-[(E)-2-phenylethenyl]phenyl}sulfanyl)acetamide
8-{2-[(4-methoxyphenyl)amino]-2-methylpropanoyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-cyclopentyl-3-phenyl-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-1H-pyrazole-5-carboxamide
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
1,5-dimethyl-4-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-acetyl-N-[2-(3,4-dimethylphenoxy)ethyl]-1H-pyrazole-5-carboxamide
2-cyclopropyl-4-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
3-{4-[1-(carbamoylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propanoic acid
(4aS,8aR)-6-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-1-propyl-decahydro-1,6-naphthyridin-2-one
2-(2,4-dimethoxyphenyl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
3-{2-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-(1-cycloheptylpiperidin-3-yl)-4-methyl-1,3-thiazole-5-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-[(propylamino)methyl]piperidin-2-one
5-cyclopropanecarbonyl-1'-(2,4-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
[3-(furan-3-carbonyl)-9-(1H-imidazol-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
3-[(dimethylamino)methyl]-1-(2,6-dimethylpyridine-4-carbonyl)pyrrolidin-3-ol
N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
N-(1-benzothiophen-2-ylmethyl)-1-cyclopropyl-N-methyl-5-oxopyrrolidine-3-carboxamide
1-(azepan-1-yl)-2-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]ethane-1,2-dione
N-{1-[(2-chlorophenyl)methyl]-1H-pyrazol-5-yl}-2-(2-hydroxyethyl)-3-oxopiperazine-1-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]benzamide
1-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-3-(methoxymethyl)pyrrolidine
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(3-methoxyphenyl)methyl]amine
N-cycloheptyl-4-oxo-1-(propan-2-yl)-5-(thiomorpholine-4-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-({5-[(3-chloro-2-fluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
5-fluoro-3-methyl-2-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indole
(1S,5R)-3-[3-(1H-pyrazol-1-yl)propanoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-tert-butyl-4-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
2-[5-(5-chloro-6-oxo-1,6-dihydropyridin-3-yl)-1-(3-fluorophenyl)-1H-1,2,4-triazol-3-yl]acetamide
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,6-dichlorobenzamide
N,N-diethyl-2-{4-[2-(2-methoxyethyl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-azaspiro[5.5]undecan-9-amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(4-methylpiperazin-1-yl)benzamide
5-propyl-4-(4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)pyrimidine
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
6-(3-fluorophenyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-chloro-N-[(1-ethylpyrrolidin-2-yl)methyl]-3-fluoro-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}benzamide
N-cyclooctyl-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
(2-methoxyethyl)[(4-methylphenyl)methyl]{[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
N-(propan-2-yl)-2-{4-[1-(propan-2-yl)piperidine-4-carbonyl]piperazin-1-yl}acetamide
2-[(5-{[benzyl(methyl)amino]methyl}-1,2-oxazol-3-yl)formamido]-N-methylbutanamide