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3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(trimethyl-1H-pyrazol-4-yl)benzamide
N-(1-cycloheptylpiperidin-3-yl)-3-acetamidobenzamide
6-(2-chlorophenyl)-N-(4-hydroxybutan-2-yl)-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(2,4-dichlorophenoxy)-1-[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrol-1-yl]ethan-1-one
[2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)phenyl]methanamine
methyl 1-[2-(cyclohexylcarbamoyl)ethyl]piperidine-2-carboxylate
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4,4-difluoropiperidine
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-[(2-chloro-6-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
3-(pentan-2-yl)-8-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-methyl-2-{2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]ethyl}-6-(trifluoromethyl)pyrimidine
N-(1-{2-[(prop-2-en-1-yl)amino]benzoyl}piperidin-4-yl)pyrimidin-2-amine
[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amine
N-[2-(dimethylamino)ethyl]-4-methoxy-3-{[1-(3-methylbut-2-enoyl)piperidin-4-yl]oxy}benzamide
1-(2,6-dimethylpyridin-4-yl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
5-[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[(1-phenylcyclopentyl)methyl]-6-[3-(1H-pyrazol-1-yl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
(4aS,8aS)-2-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
N-(carbamoylmethyl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-N-methyl-1,3-thiazol-2-amine
2-[1-({1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]pyridine
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-4-sulfamoylbenzamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-[2-(methylsulfanyl)benzoyl]piperidine
1-({5-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
7-[(2,3-dimethoxyphenyl)methyl]-2-(1-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
2-[4-(1-benzofuran-2-ylmethyl)-1-(propan-2-yl)piperazin-2-yl]ethan-1-ol
1-[4-(ethylamino)pyrimidin-2-yl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-[(1-cyclohexylpyrrolidin-3-yl)methyl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
4-({5-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
2,6-dimethyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]pyrimidine-4-carboxamide
(2S)-2-amino-1-[(3S)-3-ethylmorpholin-4-yl]-4-(methylsulfanyl)butan-1-one
4,7-dimethyl-6-(pyrimidin-5-yl)-1,3-benzothiazol-2-amine
3-methoxy-1-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine
3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-[4-(1H-imidazol-1-yl)phenyl]-3-methylurea
3-(1-benzyl-1H-imidazol-2-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
3-(2,5-dimethoxyphenyl)-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidine
1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
1-(2-{[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
N-[3-(4-fluorophenyl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
8-(4-hydroxybutyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(2R,3R)-3-{[(2-chloropyridin-3-yl)methyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(1H-indol-3-yl)-N-(oxan-3-yl)propanamide
3-[3-(dimethylamino)propyl]-5-[1-(furan-3-carbonyl)piperidin-4-yl]-5-[(2-methylphenyl)methyl]imidazolidine-2,4-dione
3-[1-(2-methyl-1-benzofuran-5-yl)-N-(pyridin-3-ylmethyl)formamido]propanoic acid
N-[(2R,3R)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-methylbutanamide
dimethyl(2-{2-[1-(morpholine-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
2-(naphthalen-2-yloxy)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}propanamide
1-benzyl-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
8-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-methyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
(2-{2-[1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine