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1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(piperidine-1-carbonyl)piperidine
5-{[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
3-[1-(3-acetamidopropanoyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[2-(3-fluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[2-({1-[3-(3-fluorophenyl)phenyl]piperidin-4-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
2-{[2-hydroxy-4-(methylsulfanyl)butanamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-{5-[5-(ethylsulfanyl)thiophene-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-{[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
6-(2,5-dimethylfuran-3-yl)-N-methyl-7-(3-methylbut-2-en-1-yl)-N-(2-methylpropyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-ethyl-1-({4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}methyl)pyrrolidine-3-carboxamide
1-{3-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}azepan-2-one
N-methyl-2-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-N,N-dimethylacetamide
[3-(2-phenylethyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl]methanol
[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
3-(2H-1,3-benzodioxol-5-yl)-N-[(1R,3S)-3-(4-methylpiperazine-1-carbonyl)cyclopentyl]propanamide
5-cyclopropanecarbonyl-1'-(thiophene-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-({1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}methyl)-4-phenylbenzamide
[(3R,4R)-1-[(4-chlorophenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-methyl-2-[4-(2-phenylethyl)piperazin-1-yl]-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
(1R,5R)-6-(1H-indazole-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{5-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(pyridin-3-yl)propanamide
3-{1-[2-(2,5-dioxoimidazolidin-1-yl)acetyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-(thiomorpholin-4-yl)ethan-1-one
5-{[3-(3-ethylphenoxy)azetidin-1-yl]methyl}-2-methoxyphenol
3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
1-[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-phenylbutane-1,4-dione
2-fluoro-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)oxane-2-carboxamide
1-{1'-[2-(dimethylamino)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
1-[2-hydroxy-3-(4-methoxy-2-{[(3-methylbutyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
5-(2,3-dihydro-1-benzofuran-2-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}propane-1,3-diol
2-chloro-4-[1-(isoquinolin-5-yl)-1H-imidazol-2-yl]phenol
1-[2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]imidazolidin-2-one
2-(3,4-difluorophenyl)-5-propyl-2,3,4,5-tetrahydro-1,5-benzothiazepine
5-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-(2-methyl-1H-indol-3-yl)acetamide
8-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1-oxa-8-azaspiro[4.5]decane
ethyl 1-(1,3-benzothiazol-2-yl)-5-[(4-formylpiperazin-1-yl)methyl]-1H-pyrazole-4-carboxylate
methyl 5-{[(1R,3R)-3-aminocyclopentyl]carbamoyl}-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxylate
[(4-fluorophenyl)methyl](methyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
3-({1,9-dioxaspiro[5.5]undecan-4-yl}sulfamoyl)-N,N-dimethylbenzamide
2-(3-fluorophenyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidine
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-(2-methylpropyl)piperidine