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4-[(2-chloro-4-fluorophenyl)methyl]-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one
7-(cyclobutylmethyl)-2-[3-(1H-pyrazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-fluoro-5-(3-phenoxypropyl)benzamide
N-ethyl-N-(pyridin-4-ylmethyl)-1-(1,3-thiazol-2-ylmethyl)piperidin-3-amine
6-cyclopropyl-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidin-4-amine
5-(4-chlorophenyl)-N-[(6-methylpyridin-2-yl)methyl]-1,2,4-triazin-3-amine
ethyl 4-(6-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-6-azaspiro[2.5]octane-1-carbonyl)piperazine-1-carboxylate
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}thiophene-2-sulfonamide
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
3-ethyl-1-[4-(4-fluorophenyl)-4-oxobutanoyl]piperidine-3-carboxylic acid
4-[(2-chlorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
butyl 4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxylate
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-cycloheptyl-2-phenylacetamide
1-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-4-(oxolane-2-carbonyl)-1,4-diazepane
1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
methyl[(3-methylpyridin-2-yl)methyl]({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)amine
1-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
(3S,9aR)-3-(4-aminobutyl)-8-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-(4-oxo-4H-chromene-2-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[2-(4-chlorophenyl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-2,2-dimethyloxane-4-carboxamide
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-(4-fluorophenyl)-N-(furan-2-ylmethyl)acetamide
N-(furan-2-ylmethyl)-N,6-dimethyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidine
2-[4-(2-hydroxyphenyl)piperazin-1-yl]-2-[4-(methylsulfanyl)phenyl]acetic acid
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-2-(1-propyl-1H-pyrazol-4-yl)quinoline
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-5-cyclopropyl-1,3,4-oxadiazol-2-amine
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-chloro-5-acetamidobenzamide
1-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-(propan-2-yl)piperidine-3-carboxamide
1-(2-aminoethyl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
(3S,4S)-4-[({[4-(pyridin-2-yl)phenyl]methyl}amino)methyl]piperidin-3-ol
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,3-dimethylbenzamide
4-ethyl-6-{4-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperazin-1-yl}pyrimidine
(3S,4S)-4-(propan-2-yl)-1-{[(pyridin-2-ylmethyl)carbamoyl]methyl}pyrrolidine-3-carboxylic acid
(5S)-5-[({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]pyrrolidin-2-one
N-{[5-(1-benzofuran-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}methanesulfonamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(methylsulfanyl)pyridine-3-carboxamide
N,3-dimethyl-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}furan-2-carboxamide
(1R,5R)-N,N-dimethyl-6-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[(3-methoxyphenyl)methyl]-N-[(3-methyl-1H-indol-2-yl)methyl]piperidin-3-amine
5-ethyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyrimidin-2-amine
8-acetyl-2-[2-(2-methoxyphenoxy)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(2-methoxyphenyl)-6-[4-(piperidin-1-yl)piperidin-1-yl]pyridazine
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
2-chloro-4-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
(1S,5R)-6-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane