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5-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)quinoline
3-cyclohexyl-N-[2-(2,3-dimethoxyphenyl)ethyl]-1H-pyrazole-4-carboxamide
2-methyl-N-[(2-methylphenyl)(pyridin-4-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(1,3-thiazol-2-ylmethyl)piperidine
2-(ethylsulfanyl)-5-[1-(1H-imidazol-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]pyrimidine
4-hydroxy-N-methyl-N-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
N'-(2-ethoxyphenyl)-N-methyl-N-(1-methylpyrrolidin-3-yl)propanediamide
5-tert-butyl-4-{[(3S,4R)-3-[(dimethylcarbamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}furan-2-carboxamide
2-[4-(propan-2-yloxy)phenyl]-2-(pyrrolidin-1-yl)acetic acid
7-[(3-methylphenyl)methyl]-2-[(6-methylpyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-(1,4-dioxan-2-ylmethyl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
7-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-1-oxa-7-azaspiro[3.5]nonane
3-{[2-(furan-2-yl)phenyl]methyl}-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-(2,2-dimethylpropanoyl)-N-(5-methyl-1,2-oxazol-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpiperazine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(3,4-difluorophenyl)methyl]methylamine
3-(azepane-1-sulfonyl)-5-(4-methyl-1H-pyrazol-1-yl)benzoic acid
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-[(2,4,6-trimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(hydroxymethyl)-N-[2-(2-propoxyphenyl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
2-(2-fluorophenyl)-N-[2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]acetamide
1-[(1S,5R)-6-(2,3-difluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
methyl (2S,4R)-1-[(4-methoxy-3-methylphenyl)methyl]-4-[3-(4-methylphenyl)propanamido]pyrrolidine-2-carboxylate
N-methyl-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
6-({[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}amino)pyrazine-2-carboxamide
1-(dimethylamino)-3-[4-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)phenoxy]propan-2-ol
(1S,5R)-3-[(5-acetylthiophen-3-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-N-phenylpyrimidin-2-amine
3-(aminomethyl)-4-(3,4-dimethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(azepan-1-yl)ethyl]-6-cyano-N-ethylpyridine-3-carboxamide
ethyl 2-[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]acetate
N-[4-({methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenyl]acetamide
(3R,7S,8aS)-7-{[(3,4-difluorophenyl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(3S,4S)-1-(1-aminocyclopentanecarbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
(4S)-4-[1-(2,3-dihydro-1H-inden-5-yl)-1H-1,2,4-triazol-5-yl]-4-acetamidobutanamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
N-[(1-cyclopentylpiperidin-3-yl)methyl]-3-methyl-N-[2-(piperidin-1-yl)ethyl]butanamide
(2E)-2-methyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}but-2-enamide
7-chloro-4-[4-(morpholin-4-ylmethyl)piperidin-1-yl]quinoline
1-ethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[(2-hydroxyethyl)sulfanyl]-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
N-cyclohexyl-N-methyl-3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-2-amine
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(2-methoxyphenyl)acetamide
4-[6-(3,4,5-trifluorophenyl)pyridine-3-carbonyl]morpholine
1-(4-fluorophenyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}cyclopropane-1-carboxamide
N,1-dimethyl-5-[methyl(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-phenyl-N-(propan-2-yl)-N-[(2,4,5-trimethoxyphenyl)methyl]acetamide
3-[(2-methylpyrrolidin-1-yl)sulfonyl]-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
4-{1-[1-(2-methylpropanoyl)piperidin-4-yl]pyrrolidin-3-yl}benzoic acid